SCHEMBL7302960

SCHEMBL7302960

CCCc1nc2ccc(-c3cn4cc(C(N)=O)ccc4n3)cc2n1Cc1ccc(-c2ccccc2C(=O)O)cc1

nearest known ligand 0.68

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PPARG P37231 16/20 0.68
AGTR1 P30556 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302965 0.90 PPARG (0.54) PPARGAGTR1
SCHEMBL682604 0.88 PPARG (0.71) PPARG
SCHEMBL7301049 0.88 AGTR1 (0.68) PPARGAGTR1
SCHEMBL7302124 0.85 PPARG (0.70) PPARGAGTR1
SCHEMBL7301700 0.83 AGTR1 (0.69) PPARGAGTR1
SCHEMBL8394674 0.83 AGTR1 (0.79) PPARGAGTR1
SCHEMBL7302715 0.83 PPARG (0.68) PPARG
SCHEMBL7302673 0.82 AGTR1 (0.56) PPARGAGTR1
SCHEMBL7310732 0.82 PPARG (0.69) PPARG
SCHEMBL7301790 0.82 PPARG (0.71) PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614519-A (1-(2,3 or 4-N-morpholinoalkyl)-imidazol-4-yl)-benizimidazol-1-yl-methyl]-biphenyls useful as angiotensin-II antagonists KARL THOMAE GMBH (DE) 1997-03-25 US disclosed
US-5602127-A ADMINISTERING TO TREAT HYPERTENSION KARL THOMAE GMBH (DE) 1997-02-11 US disclosed
US-5594003-A HYPOTENSIVE AGENTS DR. KARL THOMAE GMBH (DE) 1997-01-14 US disclosed
US-5591762-A HYPOTENSIVE AGENTS DR. KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
EP-0502314-A1 Benzimidazol, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-09 EP disclosed