SCHEMBL7302963

SCHEMBL7302963

CS(=O)(=O)Nc1ccc(N2CCC(=O)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
MAPT P10636 4/20 0.46
RECQL P46063 1/20 0.46
ADRB1 P08588 4/20 0.45
ADRB2 P07550 3/20 0.45
ADRB3 P13945 3/20 0.45
JAK2 O60674 2/20 0.45
JAK3 P52333 2/20 0.45
LMNA P02545 2/20 0.44
HPGD P15428 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
USP2 O75604 1/20 0.44
KEAP1 Q14145 1/20 0.44
KCNH2 Q12809 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824858 0.84 MAPT (0.60) ALDH1A1MAPTRECQLLMNAHPGD
SCHEMBL16261606 0.83 MAPT (0.63) ALDH1A1MAPTRECQLLMNAHPGD
SCHEMBL10426116 0.81 ALDH1A1 (0.59) ALDH1A1MAPTADRB1ADRB2ADRB3
Hydrochloric Acid SCHEMBL10426727 0.80 ALDH1A1 (0.58) ALDH1A1MAPTADRB1ADRB2ADRB3
SCHEMBL7460280 0.80 JAK2 (0.48) ALDH1A1MAPTRECQLADRB1ADRB2
SCHEMBL5851742 0.80 HTR6 (0.64) ALDH1A1ADRB1LMNAKDM4EHTR6
SCHEMBL13105531 0.79 MAPT (0.43) ALDH1A1MAPTRECQLLMNAKDM4E
Hydrochloric Acid SCHEMBL7001932 0.79 HTR6 (0.62) ALDH1A1ADRB1LMNAKDM4EHTR6
SCHEMBL10680323 0.79 JAK2 (0.50) ALDH1A1MAPTRECQLADRB1ADRB2
SCHEMBL7301452 0.78 JAK2 (0.64) ALDH1A1MAPTRECQLADRB1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481299-B1 N-phenyl-piperidyl-4-amines and drugs containing them BASF AG (DE) 1994-07-20 EP disclosed
US-5260318-A Phenylpiperidylamines and drugs containing them BASF AKTIENGESELLSCHAFT (DE) 1993-11-09 US disclosed
EP-0481299-A2 N-phenyl-piperidyl-4-amines and drugs containing them BASF Aktiengesellschaft (DE) 1992-04-22 EP disclosed