SCHEMBL7303064

SCHEMBL7303064

COc1ccc(-c2nn[c]o2)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.55
MAPK1 P28482 5/20 0.55
HPGD P15428 5/20 0.55
KDM4E B2RXH2 9/20 0.54
NPC1 O15118 8/20 0.54
SMN1; SMN2 Q16637 7/20 0.54
RAB9A P51151 5/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
HSD17B10 Q99714 6/20 0.48
MAPT P10636 2/20 0.48
PRNP P04156 1/20 0.48
ALPG P10696 1/20 0.48
PDE4A P27815 1/20 0.47
TP53 P04637 1/20 0.47
ACHE P22303 1/20 0.45
TSHR P16473 2/20 0.44
ALOX5 P09917 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23115547 0.79 TLR8 (0.65)
SCHEMBL23115488 0.79 TLR8 (0.70)
SCHEMBL345944 0.77 NPC1 (0.51) ALDH1A1HPGDKDM4ENPC1SMN1; SMN2
SCHEMBL12964716 0.77 KDM4E (0.83) ALDH1A1MAPK1HPGDKDM4ENPC1
SCHEMBL3621429 0.75 NOTUM (0.56) ALDH1A1MAPK1HPGDKDM4ENPC1
SCHEMBL7310699 0.74 ALDH1A1 (0.55) ALDH1A1MAPK1HPGDKDM4ESMN1; SMN2
SCHEMBL7312332 0.74 RAB9A (0.41) ALDH1A1HPGDKDM4ENPC1SMN1; SMN2
SCHEMBL12626897 0.74 NPC1 (0.84) ALDH1A1MAPK1HPGDKDM4ENPC1
SCHEMBL2750427 0.73 ALDH1A1 (0.51) ALDH1A1MAPK1HPGDKDM4ENPC1
SCHEMBL3613332 0.71 ALDH1A1 (0.46) ALDH1A1MAPK1HPGDKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5371074-A Use of saccharin derivatives as proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1994-12-06 US claimed
EP-0542372-A1 2-Substituted saccharin derivative proteolytic enzyme inhibitors STERLING WINTHROP INC. (US) 1993-05-19 EP claimed