SCHEMBL7303099

SCHEMBL7303099

COc1ccc(-c2csc3nc(N4CCN(c5cccc(C(F)(F)F)c5)CC4)c4cccn4c23)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.81
HTR1A P08908 7/20 0.81
TSHR P16473 4/20 0.45
MAPT P10636 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
HSD17B10 Q99714 3/20 0.43
LMNA P02545 2/20 0.43
GAA P10253 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TP53 P04637 2/20 0.42
KDM4E B2RXH2 2/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
NFKB1 P19838 1/20 0.42
HTR1D P28221 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303643 0.90 HTR2C (1.00) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL7296642 0.75 HTR2C (1.00) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL7298654 0.74 HTR2C (0.86) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL7298088 0.74 HTR2C (1.00) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL8567807 0.71 HTR2C (0.72) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL7298486 0.71 HTR2C (1.00) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL7296823 0.68 HTR2C (0.75) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL8880281 0.67 HTR2C (0.66) HTR2CHTR1ATSHRMAPTSMN1; SMN2
SCHEMBL7303868 0.67 HTR1A (1.00) HTR2CHTR1AHTR3EHTR3BHTR3A
SCHEMBL7302481 0.64 HTR1A (0.74) HTR2CHTR1AHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573360-B1 Pyrrolothienopyrazine compounds as 5-HT3 receptors antagonists ADIR (FR) 1998-08-26 EP disclosed
EP-0573360-A1 Pyrrolothienopyrazine compounds as 5-HT3 receptors antagonists ADIR ET COMPAGNIE (FR) 1993-12-08 EP disclosed