SCHEMBL7303316

SCHEMBL7303316

O=c1[nH]c(=O)n(CCCCN2CC=C(c3ccccc3)CC2)c2cc(O)c(O)cc12

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 16/20 0.64
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
HTR1A P08908 1/20 0.48
MAPT P10636 1/20 0.48
CYP2C9 P11712 1/20 0.48
DRD2 P14416 1/20 0.48
TSHR P16473 1/20 0.48
DRD4 P21917 1/20 0.48
CYP2C19 P33261 1/20 0.48
DRD3 P35462 1/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7303725 0.99 PARP1 (0.63) PARP1CYP1A2CYP3A4HTR1AMAPT
SCHEMBL7307656 0.89 PARP1 (0.63) PARP1CYP1A2CYP3A4HTR1AMAPT
Bromide SCHEMBL7301782 0.88 PARP1 (0.62) PARP1CYP1A2CYP3A4HTR1AMAPT
Bromide SCHEMBL7309634 0.88 PARP1 (0.62) PARP1CYP1A2CYP3A4HTR1AMAPT
SCHEMBL7305161 0.86 PARP1 (0.73) PARP1
SCHEMBL7308205 0.85 PARP1 (0.64) PARP1HTR1AMAPTTSHRTDP1
SCHEMBL7308221 0.85 PARP1 (0.63) PARP1
SCHEMBL7302855 0.85 PARP1 (0.64) PARP1DRD2
Hydrochloric Acid SCHEMBL7301544 0.85 PARP1 (0.63) PARP1MAPT
Hydrochloric Acid SCHEMBL7301868 0.84 PARP1 (0.62) PARP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5304560-A Treating CNS disorders; dopamine receptor antagonist FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-19 US claimed
EP-0481342-A1 Quinazoline derivatives and their preparation FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-04-22 EP claimed