SCHEMBL730382

SCHEMBL730382

OCC#Cc1cccc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
MAPT P10636 2/20 0.48
MITF O75030 1/20 0.48
HTT P42858 1/20 0.48
RAD52 P43351 1/20 0.48
CHAT P28329 1/20 0.45
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 2/20 0.44
POLB P06746 1/20 0.44
GRM5 P41594 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP2A6 P11509 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
ACACB O00763 1/20 0.40
ALOX15 P16050 1/20 0.38
HRH3 Q9Y5N1 4/20 0.38
TDP1 Q9NUW8 2/20 0.37
TSHR P16473 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9274173 0.87 ALDH1A1 (0.36) MEN1KMT2AMAPTMITFHTT
SCHEMBL2410459 0.82 MAPT (0.54) MEN1KMT2AMAPTMITFHTT
SCHEMBL31323032 0.80 CYP1A2 (0.38) MEN1KMT2AMAPTMITFHTT
SCHEMBL6449051 0.80 CYP1A2 (0.44) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL29661843 0.80 CHAT (0.60) MEN1KMT2AMAPTMITFHTT
SCHEMBL30515632 0.80 CYP1A2 (0.44) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL2776015 0.80 CHAT (0.60) MEN1KMT2AMAPTMITFHTT
SCHEMBL1858300 0.80 MEN1 (0.48) MEN1KMT2AMAPTMITFHTT
SCHEMBL7573003 0.80 MEN1 (0.48) MEN1KMT2AMAPTMITFHTT
SCHEMBL27481040 0.80 CHAT (0.49) MEN1KMT2AMAPTMITFHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103570489-B Method for preparing cis-olefin from alkyne through copper catalysis UNIV NORTHWEST A&F 2015-06-24 CN claimed
CN-103570489-A Method for preparing cis-olefin from alkyne through copper catalysis UNIV NORTHWEST A&F 2014-02-12 CN claimed
US-5399676-A DNA sequence identification GILEAD SCIENCES (US) 1995-03-21 US claimed
US-11814462-B2 Functionalized cyclic polymers and methods of preparing same UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2023-11-14 US disclosed
US-20220056167-A1 Functionalized Cyclic Polymers and Methods of Preparing Same NATIONAL SCIENCE FOUNDATION 2022-02-24 US disclosed
WO-2020223672-A1 FUNCTIONALIZED CYCLIC POLYMERS AND METHODS OF PREPARING SAME UNIVERSITY OF FLORIDA RESEARCHFOUNDATION, INC. (US) 2020-11-05 WO disclosed
CN-103570489-B Method for preparing cis-olefin from alkyne through copper catalysis UNIV NORTHWEST A&F 2015-06-24 CN disclosed
CN-103570489-A Method for preparing cis-olefin from alkyne through copper catalysis UNIV NORTHWEST A&F 2014-02-12 CN disclosed
US-8138377-B2 Arylbicyclo[3.1.0]hexylamines and methods and compositions for their preparation and use DOV PHARMACEUTICAL, INC. (US) 2012-03-20 US disclosed
US-8138377-B2 Arylbicyclo[3.1.0]hexylamines and methods and compositions for their preparation and use DOV PHARMACEUTICAL, INC. (US) 2012-03-20 US disclosed
US-20110105544-A1 CARBOXYLIC DERIVATIVES FOR USE IN THE TREATMENT OF CANCER CRYSTAX PHARMACEUTICALS, S.L. (ES) 2011-05-05 US disclosed
WO-2009080722-A2 CARBOXYLIC DERIVATIVES FOR USE IN THE TREATMENT OF CANCER CRYSTAX PHARMACEUTICALS, S.L. (ES) 2009-07-02 WO disclosed
US-20080293822-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use ETHISMOS RESEARCH, INC. 2008-11-27 US disclosed
US-20080293822-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use ETHISMOS RESEARCH, INC. 2008-11-27 US disclosed
US-20080269348-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use ETHISMOS RESEARCH, INC. 2008-10-30 US disclosed
US-20080269348-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use ETHISMOS RESEARCH, INC. 2008-10-30 US disclosed
US-20080194696-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use ETHISMOS RESEARCH, INC. 2008-08-14 US disclosed
US-20080194696-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use ETHISMOS RESEARCH, INC. 2008-08-14 US disclosed
WO-2008057575-A2 NOVEL ARYLBICYCLO[3.1.0]HEXYLAMINES AND METHODS AND COMPOSITIONS FOR THEIR PREPARATION AND USE DOV PHARMACEUTICAL, INC. (US) 2008-05-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080194696-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use HTR2C, HTR1B, HTR3C MEN1 1876/4885KMT2A 415/4885MAPT 274/4885
US-20080293822-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use HTR2C, HTR1B, HTR3C MEN1 1876/4885KMT2A 415/4885MAPT 274/4885
US-20080269348-A1 Novel Arylbicyclo[3.1.0]Hexylamines And Methods And Compositions For Their Preparation And Use HTR2C, HTR1B, HTR3C MEN1 1876/4885KMT2A 415/4885MAPT 274/4885
US-20110105544-A1 CARBOXYLIC DERIVATIVES FOR USE IN THE TREATMENT OF CANCER AKR1C3, TPD52L2, HCCS MEN1 1865/4885KMT2A 2127/4885MAPT 4342/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.