SCHEMBL7303829

SCHEMBL7303829

COC(=O)CCN1CCN(CC2CN(C3CCN(C(C)C)CC3)C(=O)O2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 5/20 0.47
SMN1; SMN2 Q16637 1/20 0.39
TP53 P04637 1/20 0.35
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRL1 P41146 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HTR4 Q13639 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.32
HRH3 Q9Y5N1 2/20 0.32
SIGMAR1 Q99720 2/20 0.32
PARP1 P09874 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
SLC5A7 Q9GZV3 1/20 0.31
CCR2 P41597 1/20 0.31
KCNH2 Q12809 1/20 0.31
BCHE P06276 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314554 0.94 HTR2B (0.45) HTR2BSMN1; SMN2OPRM1OPRD1OPRL1
SCHEMBL7302525 0.90 HTR2B (0.48) HTR2BOPRM1OPRD1OPRL1ITGB3
SCHEMBL7311678 0.89 HTR2B (0.45) HTR2BSMN1; SMN2TP53OPRM1OPRD1
SCHEMBL7310988 0.89 HTR2B (0.52) HTR2BHTR4PARP1PARP2CCR2
SCHEMBL7304864 0.85 HTR2B (0.43) HTR2BSMN1; SMN2TP53ITGB3ITGA2B
SCHEMBL7314426 0.84 HTR2B (0.50) HTR2BSMN1; SMN2HTR4PARP1PARP2
SCHEMBL7309599 0.84 SMN1; SMN2 (0.42) HTR2BSMN1; SMN2TP53OPRM1OPRD1
SCHEMBL7311014 0.83 HTR2B (0.43) HTR2BSMN1; SMN2TP53ITGB3ITGA2B
SCHEMBL7309942 0.83 SMN1; SMN2 (0.37) HTR2BSMN1; SMN2TP53OPRM1OPRD1
SCHEMBL7316422 0.82 HTR2B (0.40) HTR2BSMN1; SMN2TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed