SCHEMBL7302525

SCHEMBL7302525

COC(=O)CN1CCN(CC2CN(C3CCN(C(C)C)CC3)C(=O)O2)CC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 6/20 0.48
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
HRH3 Q9Y5N1 3/20 0.34
SIGMAR1 Q99720 5/20 0.32
PARP1 P09874 1/20 0.32
PARP2 Q9UGN5 1/20 0.32
CCR2 P41597 1/20 0.32
KCNH2 Q12809 1/20 0.32
P2RX3 P56373 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRL1 P41146 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303829 0.90 HTR2B (0.47) HTR2BITGB3ITGA2BHRH3SIGMAR1
SCHEMBL7307896 0.88 HTR2B (0.46) HTR2BITGB3ITGA2BHRH3SIGMAR1
SCHEMBL7308689 0.88 HTR2B (0.54) HTR2BITGB3ITGA2BHRH3SIGMAR1
SCHEMBL7314554 0.88 HTR2B (0.45) HTR2BITGB3ITGA2BHRH3CCR2
SCHEMBL7313313 0.85 HTR2B (0.45) HTR2BITGB3ITGA2BSIGMAR1OPRL1
SCHEMBL7318339 0.83 ITGB3 (0.45) HTR2BITGB3ITGA2BSIGMAR1OPRM1
SCHEMBL7310988 0.82 HTR2B (0.52) HTR2BPARP1PARP2CCR2KCNH2
SCHEMBL7314767 0.82 ITGB3 (0.38) HTR2BITGB3ITGA2BHRH3CCR2
SCHEMBL7309068 0.82 HTR2B (0.41) HTR2BITGB3ITGA2B
SCHEMBL7303558 0.81 HTR2B (0.52) HTR2BITGB3ITGA2BSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed