SCHEMBL7314554

SCHEMBL7314554

COC(=O)CCCN1CCN(CC2CN(C3CCN(C(C)C)CC3)C(=O)O2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 5/20 0.45
HSD17B10 Q99714 1/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAOA P21397 1/20 0.32
HDAC1 Q13547 1/20 0.32
EHMT1 Q9H9B1 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRL1 P41146 1/20 0.32
CCR8 P51685 2/20 0.32
CCR2 P41597 1/20 0.32
KCNH2 Q12809 1/20 0.32
HTR4 Q13639 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7303829 0.94 HTR2B (0.47) HTR2BITGB3ITGA2BSMN1; SMN2OPRM1
SCHEMBL7311014 0.90 HTR2B (0.43) HTR2BHSD17B10ITGB3ITGA2BSMN1; SMN2
SCHEMBL7314426 0.89 HTR2B (0.50) HTR2BHSD17B10SMN1; SMN2MAOAHTR4
SCHEMBL7302525 0.88 HTR2B (0.48) HTR2BITGB3ITGA2BOPRM1OPRD1
SCHEMBL7310988 0.85 HTR2B (0.52) HTR2BCCR2KCNH2HTR4MEN1
SCHEMBL7310324 0.85 HTR2B (0.40) HTR2BHSD17B10ITGB3ITGA2BSMN1; SMN2
SCHEMBL7313291 0.84 HTR2B (0.40) HTR2BITGB3ITGA2BSMN1; SMN2MAOA
SCHEMBL7305668 0.84 HTR2B (0.36) HTR2BITGB3ITGA2BMAOACCR2
SCHEMBL7311678 0.83 HTR2B (0.45) HTR2BHSD17B10ITGB3ITGA2BSMN1; SMN2
SCHEMBL7306441 0.82 HTR2B (0.48) HTR2BOPRM1OPRD1CCR8LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed