SCHEMBL7304584

SCHEMBL7304584

CC(=O)SCC(Cc1ccccc1)NC(=O)NCCC(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MME P08473 3/20 0.46
ACE P12821 2/20 0.46
MEN1 O00255 1/20 0.45
TSHR P16473 1/20 0.45
KMT2A Q03164 1/20 0.45
MMEL1 Q495T6 1/20 0.45
NAALAD2 Q9Y3Q0 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ABCC3 O15438 1/20 0.44
NR1I2 O75469 1/20 0.44
ABCB11 O95342 1/20 0.44
NR3C1 P04150 1/20 0.44
RARG P13631 1/20 0.44
CNR1 P21554 1/20 0.44
OPRK1 P41145 1/20 0.44
NR1H2 P55055 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9587977 0.89 KMT2A (0.59) MMEMEN1TSHRKMT2AOPRK1
SCHEMBL7298881 0.87 MME (0.58) MMEACEMEN1KMT2AMMEL1
SCHEMBL9587602 0.83 MME (0.48) MMEACECYP1A2CYP3A4CYP2D6
SCHEMBL9588619 0.81 CYP3A4 (0.54) MMEKMT2AMMEL1CYP1A2CYP3A4
SCHEMBL9068906 0.81 MME (0.54) MMEACE
SCHEMBL9068533 0.80 MME (0.62) MMEACECYP3A4
SCHEMBL9588091 0.80 MME (0.62) MMEACE
SCHEMBL9068556 0.80 MME (0.53) MMEACE
SCHEMBL9588793 0.80 CYP3A4 (0.46) MMEACECYP1A2CYP3A4CYP2D6
SCHEMBL7276817 0.80 ACE (0.65) MMEACEMMEL1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0465369-B1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1994-04-13 EP disclosed
US-5190974-A Analgesics ROUSSEL UCLAF (FR) 1993-03-02 US disclosed
EP-0465369-A1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1992-01-08 EP disclosed