SCHEMBL7305076

SCHEMBL7305076

C=CCOc1ccc(-c2ccncc2)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.43
MAPT P10636 2/20 0.43
GCGR P47871 1/20 0.38
MAPK14 Q16539 1/20 0.38
ELOVL1 Q9BW60 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
CYP2A6 P11509 1/20 0.35
AURKA O14965 1/20 0.34
TTK P33981 1/20 0.34
AURKB Q96GD4 1/20 0.34
INCENP Q9NQS7 1/20 0.34
SNCA P37840 1/20 0.34
PIK3CA P42336 1/20 0.34
CDK2 P24941 1/20 0.34
GSK3B P49841 1/20 0.34
MKNK1 Q9BUB5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7278725 0.77 CYP19A1 (0.64) CYP19A1MAPTELOVL1CYP3A4CYP2D6
SCHEMBL3824432 0.73 CA12 (0.44) MAPTCYP2D6KDM4EALDH1A1LMNA
SCHEMBL8027259 0.73 KDM4E (0.38) MAPTKDM4EALDH1A1SNCAMAPK1
SCHEMBL1422827 0.73 CYP19A1 (0.62) CYP19A1MAPTCYP2A6AURKATTK
SCHEMBL6213208 0.72 KDM4E (0.43) MAPTKDM4EALDH1A1CDK2MAPK1
SCHEMBL5762848 0.72 TSHR (0.41) MAPTGCGRMAPK14KDM4EALDH1A1
SCHEMBL13764327 0.70 CA12 (0.48) MAPTCYP2D6KDM4EALDH1A1LMNA
SCHEMBL12380456 0.69 ALDH1A1 (0.39) MAPTCYP2D6KDM4EALDH1A1LMNA
SCHEMBL3260151 0.67 CHRNB2 (0.44) MAPTCYP2D6KDM4EALDH1A1LMNA
SCHEMBL10517456 0.67 SMN1; SMN2 (0.47) MAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0200024-B1 3-CYANO-PYRIDINES, PROCESS FOR THEIR PREPARATION AND THEIR PHARMACEUTICAL USE ARZNEIMITTELWERK DRESDEN GmbH (DE) 1992-07-01 EP disclosed
EP-0200024-A2 3-Cyano-pyridines, process for their preparation and their pharmaceutical use ARZNEIMITTELWERK DRESDEN GmbH (DE) 1986-11-05 EP disclosed