SCHEMBL7306441

SCHEMBL7306441

COC(=O)CCCN1CCN(CC2CN(C3CCN(Cc4ccccc4)CC3)C(=O)O2)CC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 3/20 0.48
CCR8 P51685 2/20 0.44
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
CHRM2 P08172 3/20 0.41
CHRM3 P20309 3/20 0.41
CACNA1G O43497 1/20 0.41
SIGMAR1 Q99720 3/20 0.41
TMEM97 Q5BJF2 1/20 0.41
HTR1A P08908 1/20 0.40
LMNA P02545 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
TSHR P16473 1/20 0.40
ABCB1 P08183 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307163 0.95 HTR2B (0.50) HTR2BCCR8CYP2D6CYP2C9ALDH1A1
SCHEMBL7306400 0.90 HTR2B (0.53) HTR2BCCR8CYP2D6CYP2C9CHRM2
SCHEMBL7303558 0.89 HTR2B (0.52) HTR2BCCR8ALDH1A1CHRM2CHRM3
SCHEMBL7307261 0.87 ALDH1A1 (0.41) ALDH1A1MAPTCACNA1GSIGMAR1TMEM97
SCHEMBL7314325 0.86 ALDH1A1 (0.43) ALDH1A1MAPTCACNA1GSIGMAR1TMEM97
SCHEMBL7310156 0.86 ALDH1A1 (0.43) ALDH1A1MAPTCACNA1GSIGMAR1TMEM97
SCHEMBL7314130 0.86 ALDH1A1 (0.43) HTR2BALDH1A1MAPTCACNA1GSIGMAR1
SCHEMBL7305773 0.86 HTR2B (0.54) HTR2BCCR8CYP2D6CYP2C9CHRM2
SCHEMBL7311014 0.86 HTR2B (0.43) HTR2BCCR8ALDH1A1SIGMAR1LMNA
SCHEMBL7303582 0.85 ACHE (0.45) ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed