SCHEMBL7306016

SCHEMBL7306016

O=C1CNC(c2ccccc2)C(c2ccccc2)O1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
GRM5 P41594 1/20 0.39
GBA1 P04062 1/20 0.38
CA2 P00918 1/20 0.38
GAA P10253 2/20 0.37
ALDH1A1 P00352 2/20 0.36
SLC6A2 P23975 1/20 0.36
ADRA1A P35348 1/20 0.36
HTR2B P41595 1/20 0.36
SLC6A3 Q01959 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ADORA3 P0DMS8 1/20 0.35
AR P10275 1/20 0.35
CYP19A1 P11511 1/20 0.35
MAOB P27338 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3706077 1.00 CYP2C9 (0.42) CYP2C9CYP2C19SMN1; SMN2GRM5GBA1
SCHEMBL249120 1.00 CYP2C9 (0.42) CYP2C9CYP2C19SMN1; SMN2GRM5GBA1
SCHEMBL12525029 1.00 CYP2C9 (0.42) CYP2C9CYP2C19SMN1; SMN2GRM5GBA1
SCHEMBL12524998 1.00 CYP2C9 (0.42) CYP2C9CYP2C19SMN1; SMN2GRM5GBA1
SCHEMBL14980914 0.82 SMN1; SMN2 (0.38) CYP2C9CYP2C19SMN1; SMN2GBA1CA2
SCHEMBL23841973 0.80 CYP2C9 (0.41) CYP2C9CYP2C19CA2GAAALDH1A1
SCHEMBL135940 0.77 CA2 (0.40) CYP2C9CYP2C19SMN1; SMN2CA2GAA
SCHEMBL1443275 0.71 GRM5 (0.66) SMN1; SMN2GRM5CA2
SCHEMBL14508491 0.71 GRM5 (0.66) SMN1; SMN2GRM5CA2
SCHEMBL2798313 0.71 GRM5 (0.66) SMN1; SMN2GRM5CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106147887-B Methanol gasoline multiphase corrosion inhibitor and methanol gasoline prepared from same 福建中源新能源股份有限公司 2018-05-04 CN claimed
CN-106147887-A Methanol gasoline multiphase corrosion inhibitor and methanol gasoline prepared from same 福建中源新能源股份有限公司 2016-11-23 CN claimed
US-11932624-B2 MDM2 degraders and uses thereof KYMERA THERAPEUTICS, INC. (US) 2024-03-19 US disclosed
US-20240025878-A1 MDM2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. 2024-01-25 US disclosed
US-20230233546-A1 METHODS OF TREATING CANCER KYMERA THERAPEUTICS, INC. 2023-07-27 US disclosed
WO-2023114933-A1 METHODS OF TREATING CANCER KYMERA THERAPEUTICS, INC. (US) 2023-06-22 WO disclosed
WO-2023049790-A2 MDM2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2023-03-30 WO disclosed
CN-115776887-A MDM2 degrading agents and uses thereof 凯麦拉医疗公司 2023-03-10 CN disclosed
EP-4121043-A1 MDM2 DEGRADERS AND USES THEREOF Kymera Therapeutics, Inc. (US) 2023-01-25 EP disclosed
WO-2021188948-A1 MDM2 DEGRADERS AND USES THEREOF KYMERA THERAPEUTICS, INC. (US) 2021-09-23 WO disclosed
CN-105189524-B The synthetic method of optical activity alpha-amino acid 浜理药品工业株式会社 2019-07-19 CN disclosed
EP-0592367-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1994-04-13 EP disclosed
WO-1994005677-A1 PHOSPHONO SUBSTITUTED TETRAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1994-03-17 WO disclosed
US-5294632-A Diuretics and vasorelaxants CIBA-GEIGY CORPORATION (US) 1994-03-15 US disclosed
US-5273990-A 5-Phosphonomethyleneamino aryl-substitued alkylene-1H-tetazoles CIBA-GEIGY CORPORATION (US) 1993-12-28 US disclosed
US-5250522-A Neutral endopeptidase inhibitors; cardiovascular disorders CIBA-GEIGY CORPORATION (US) 1993-10-05 US disclosed
EP-0555175-A1 Biaryl substituted 4-amino-butyric acid amides CIBA-GEIGY AG (CH) 1993-08-11 EP disclosed
US-5217996-A Endopeptidase inhibitors CIBA-GEIGY CORPORATION (US) 1993-06-08 US disclosed
EP-0511940-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1992-11-04 EP disclosed
US-5155100-A Treating cardiovascular disorders in mammals CIBA-GEIGY CORPORATION (US) 1992-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230233546-A1 METHODS OF TREATING CANCER TP53, MDM2, MCL1 CYP2C9 3919/4885CYP2C19 3827/4885SMN1; SMN2 1499/4885
US-20240025878-A1 MDM2 DEGRADERS AND USES THEREOF MDM2, TP53, MDM4 CYP2C9 2267/4885CYP2C19 2181/4885SMN1; SMN2 3149/4885
US-11932624-B2 MDM2 degraders and uses thereof MDM2, TP53, MDM4 CYP2C9 2267/4885CYP2C19 2181/4885SMN1; SMN2 3149/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.