SCHEMBL7306027

SCHEMBL7306027

N#Cc1c([O])ccc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
ALDH1A1 P00352 6/20 0.45
KDM4E B2RXH2 4/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 1/20 0.45
MEN1 O00255 2/20 0.45
GAA P10253 2/20 0.45
MAPT P10636 2/20 0.45
KMT2A Q03164 2/20 0.45
CYP3A4 P08684 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 2/20 0.44
CYP2A6 P11509 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
CACNA1B Q00975 1/20 0.43
APBA1 Q02410 1/20 0.43
HPRT1 P00492 1/20 0.41
PAX8 Q06710 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5251870 0.79 CYP1A2 (0.54) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL646163 0.77 CA1 (0.52) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL6235233 0.75 ALDH1A1 (0.45) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL50873 0.75 ALDH1A1 (0.45) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL8331897 0.75 CYP2A6 (0.54) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL1392608 0.75 ALDH1A1 (0.45) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL5251868 0.75 ALDH1A1 (0.48) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL1855575 0.75 ESR1 (0.54) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL2419451 0.75 ALDH1A1 (0.46) CA1CA2ALDH1A1KDM4ECYP1A2
SCHEMBL16936582 0.75 ALDH1A1 (0.45) CA1CA2ALDH1A1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5629406-A AMINO ACID DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1997-05-13 US disclosed
EP-0587311-A1 Peptides capable of inhibiting the activity of HIV protease, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed