SCHEMBL7306722

SCHEMBL7306722

O=C(O)c1ccc(NC(=O)[C@H](Cc2ccc(-c3ccccc3)cc2)N(CP(=O)(O)O)c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.46
ALDH1A1 P00352 2/20 0.42
KMT2A Q03164 2/20 0.42
PKM P14618 1/20 0.42
CRHBP P24387 1/20 0.42
RAB9A P51151 1/20 0.42
CRHR2 Q13324 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
EPHX2 P34913 1/20 0.42
ADCY6 O43306 1/20 0.41
ADCY3 O60266 1/20 0.41
ADCY9 O60503 1/20 0.41
ADCY5 O95622 1/20 0.41
ADCY8 P40145 1/20 0.41
GCGR P47871 1/20 0.41
ADCY7 P51828 1/20 0.41
ADCY2 Q08462 1/20 0.41
ADCY1 Q08828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7315627 0.83 ACP3 (0.43) NR1H4ALDH1A1KMT2APKMCRHBP
SCHEMBL7308016 0.81 ALDH1A1 (0.45) NR1H4ALDH1A1KMT2APKMCRHBP
SCHEMBL7316590 0.79 MMEL1 (0.58)
SCHEMBL7310435 0.79 MMEL1 (0.58)
SCHEMBL7309927 0.78 MMEL1 (0.49) KMT2AADCY6ADCY3ADCY9ADCY5
SCHEMBL7322648 0.77 MMEL1 (0.50)
SCHEMBL7312117 0.77 MME (0.52) NR1H4ALDH1A1KMT2APKMCRHBP
SCHEMBL7312109 0.77 MME (0.52) NR1H4ALDH1A1KMT2APKMCRHBP
SCHEMBL7320409 0.76 MMEL1 (0.48)
SCHEMBL7317919 0.75 PPID (0.41) KMT2ARAB9ASMN1; SMN2ACP3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511940-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1992-11-04 EP claimed
EP-0592367-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1994-04-13 EP disclosed
US-5294632-A Diuretics and vasorelaxants CIBA-GEIGY CORPORATION (US) 1994-03-15 US disclosed
EP-0511940-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1992-11-04 EP disclosed
US-5155100-A Treating cardiovascular disorders in mammals CIBA-GEIGY CORPORATION (US) 1992-10-13 US disclosed