SCHEMBL7308016

SCHEMBL7308016

CC(N(C)[C@@H](Cc1ccc(-c2ccccc2)cc1)C(=O)Nc1ccc(C(=O)O)cc1)P(=O)(O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
MAPT P10636 1/20 0.45
TAAR1 Q96RJ0 1/20 0.43
KMT2A Q03164 2/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
MEN1 O00255 1/20 0.43
NR1H4 Q96RI1 2/20 0.43
ADCY6 O43306 1/20 0.43
ADCY3 O60266 1/20 0.43
ADCY9 O60503 1/20 0.43
ADCY5 O95622 1/20 0.43
ADCY8 P40145 1/20 0.43
GCGR P47871 1/20 0.43
ADCY7 P51828 1/20 0.43
ADCY2 Q08462 1/20 0.43
ADCY1 Q08828 1/20 0.43
ADCY4 Q8NFM4 1/20 0.43
MCHR1 Q99705 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343580 0.87 MCHR1 (0.42) ALDH1A1MAPTTAAR1MCHR1MME
SCHEMBL7306722 0.81 NR1H4 (0.46) ALDH1A1MAPTTAAR1KMT2AADRB1
SCHEMBL7348051 0.81 ACP3 (0.50) ALDH1A1MAPTMMEANPEP
SCHEMBL7322719 0.81 ACP3 (0.50) ALDH1A1MAPTMMEANPEP
SCHEMBL7315627 0.79 ACP3 (0.43) ALDH1A1MAPTKMT2AADRB1ADRB3
SCHEMBL7309958 0.79 MMEL1 (0.58) MME
SCHEMBL7318079 0.79 MMEL1 (0.58) MME
SCHEMBL7312117 0.77 MME (0.52) ALDH1A1KMT2AADRB1ADRB3NR1H4
SCHEMBL7312109 0.77 MME (0.52) ALDH1A1KMT2AADRB1ADRB3NR1H4
SCHEMBL7308004 0.75 USP30 (0.54) ALDH1A1TAAR1KMT2AADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0592367-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1994-04-13 EP disclosed
US-5294632-A Diuretics and vasorelaxants CIBA-GEIGY CORPORATION (US) 1994-03-15 US disclosed
EP-0511940-A2 Phosphono/biaryl substituted dipeptide derivatives CIBA-GEIGY AG (CH) 1992-11-04 EP disclosed
US-5155100-A Treating cardiovascular disorders in mammals CIBA-GEIGY CORPORATION (US) 1992-10-13 US disclosed