SCHEMBL7306942

SCHEMBL7306942

COc1ccc(OC(N)=S)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
CA12 O43570 1/20 0.52
CA7 P43166 1/20 0.52
CA9 Q16790 1/20 0.52
CA14 Q9ULX7 1/20 0.52
PARP10 Q53GL7 2/20 0.50
PRSS1 P07477 1/20 0.50
PRSS2 P07478 1/20 0.50
PRSS3 P35030 1/20 0.50
PARP1 P09874 1/20 0.50
PARP2 Q9UGN5 1/20 0.50
PARP4 Q9UKK3 1/20 0.50
NOS3 P29474 2/20 0.48
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
HTR3A P46098 1/20 0.48
HTR3D Q70Z44 1/20 0.48
HTR3C Q8WXA8 1/20 0.48
TDP1 Q9NUW8 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11485695 0.81 LMNA (0.52) CA1CA2CA9PRSS1TDP1
SCHEMBL8103773 0.80 GAA (0.47) PRSS1TDP1ALDH1A1HPGDGAA
SCHEMBL2463820 0.80 CA1 (0.58) CA1CA2CA12CA7CA9
SCHEMBL20072412 0.78 CA1 (0.55) CA1CA2CA12CA7CA9
SCHEMBL6310745 0.77 CA4 (0.42) ALDH1A1CYP3A4GAA
SCHEMBL201860 0.76 CA1 (0.61) CA1CA2CA12CA7CA9
SCHEMBL10754710 0.76 CA1 (0.52) CA1CA2CA12CA7CA9
SCHEMBL731242 0.76 CA1 (0.61) CA1CA2CA12CA7CA9
SCHEMBL28413733 0.76 CA1 (0.52) CA1CA2CA12CA7CA9
SCHEMBL29240594 0.76 MAPT (0.43) CA1CA2CA9MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114149353-B N-alkyl/N-aryl thioamide derivatives, and synthetic method and application thereof 华东师范大学 2024-05-17 CN disclosed
US-5674864-A ANALGESICS; ENDOPEPTIDASE AND ENKEPHALINASE INHIBITORS; CARDIOTONIC, PSYCHOTROPIC AND HYPERTENSIVE AGENTS ROUSSEL UCLAF (FR) 1997-10-07 US disclosed
EP-0465369-B1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL UCLAF (FR) 1994-04-13 EP disclosed
US-5190974-A Analgesics ROUSSEL UCLAF (FR) 1993-03-02 US disclosed
EP-0465369-A1 N-substituted derivatives of alpha-mercapto alkylamines, process for their preparation and intermediates obtained, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1992-01-08 EP disclosed