SCHEMBL7307136

SCHEMBL7307136

CC(C)(C)OC(=O)N(Cc1ccc(NC(=N)NC(=O)O)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
CYP17A1 P05093 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
AKT1 P31749 2/20 0.36
GRM2 Q14416 1/20 0.35
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35
BACE1 P56817 1/20 0.35
PTPN11 Q06124 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7944753 0.84 BACE1 (0.46) HDAC3HDAC1HDAC2NCOR2AKT1
SCHEMBL7958341 0.83 GRM2 (0.41) HDAC3HDAC1HDAC2NCOR2CYP17A1
SCHEMBL3819098 0.75 AKT1 (0.52) HDAC3HDAC1HDAC2NCOR2AKT1
SCHEMBL8363611 0.74 HDAC3 (0.43) HDAC3HDAC1HDAC2NCOR2AKT1
SCHEMBL5846695 0.74 HDAC1 (0.43) HDAC3HDAC1HDAC2NCOR2AKT1
SCHEMBL6792190 0.73 GRM2 (0.43) HDAC3HDAC1HDAC2NCOR2GRM2
SCHEMBL6690431 0.73 BACE1 (0.41) AKT1GRM2BACE1
SCHEMBL19153416 0.72 AKT1 (0.43) HDAC3HDAC1HDAC2NCOR2AKT1
SCHEMBL7944783 0.72 GRM2 (0.44) HDAC3HDAC1HDAC2NCOR2AKT1
SCHEMBL7307133 0.72 KIF11 (0.35) PTPN11NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1050534-B1 2,3-methano-amino acid derivatives, process for their preparation and pharmaceutical compositions containing them SERVIER LAB (FR) 2001-12-05 EP disclosed
EP-1050534-A1 2,3-methano-amino acid derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2000-11-08 EP disclosed