SCHEMBL7958341

SCHEMBL7958341

CC(C)(C)OC(=O)N(Cc1ccc(NC(=N)N)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.41
CYP17A1 P05093 1/20 0.40
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
NCOR2 Q9Y618 1/20 0.37
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36
MMP13 P45452 1/20 0.36
NAMPT P43490 2/20 0.36
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
AKT1 P31749 2/20 0.35
F2 P00734 2/20 0.35
AURKA O14965 1/20 0.35
RPS6KB1 P23443 1/20 0.35
TMPRSS6 Q8IU80 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307136 0.83 HDAC3 (0.38) GRM2CYP17A1HDAC3HDAC1HDAC2
SCHEMBL6792190 0.82 GRM2 (0.43) GRM2HDAC3HDAC1HDAC2NCOR2
SCHEMBL7317645 0.79 BCHE (0.42) BCHEACHEF2TMPRSS6PLG
SCHEMBL7944783 0.78 GRM2 (0.44) GRM2HDAC3HDAC1HDAC2NCOR2
SCHEMBL18300382 0.77 HDAC3 (0.41) GRM2HDAC3HDAC1HDAC2NCOR2
SCHEMBL5846695 0.77 HDAC1 (0.43) GRM2HDAC3HDAC1HDAC2NCOR2
SCHEMBL8363611 0.77 HDAC3 (0.43) GRM2HDAC3HDAC1HDAC2NCOR2
SCHEMBL5595635 0.77 NAMPT (0.58) CYP17A1HDAC1NAMPTAURKARPS6KB1
SCHEMBL3440346 0.77 KIF11 (0.43) CYP17A1BCHEACHENPC1
SCHEMBL7421165 0.76 MEN1 (0.39) BCHEACHEF2TMPRSS6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288077-B1 2-AZABICYCLO(3.1.0)HEXANE-1,2-DICARBOXYLIC AMIDE OR 2-AZABICYCLO(4.1.0)HEPTANE-1,2-DICARBOXYLIC AMIDE DERIVATIVE; TRYPSIN-LIKE SERINE PROTEASE INHIBITOR; ANTICOAGULANTS ADIR ET COMPAGNIE (FR) 2001-09-11 US disclosed