SCHEMBL7307307

SCHEMBL7307307

N[C@@H](Cc1cccs1)C(=O)ON1C(=O)c2ccccc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLA P06280 1/20 0.45
BRCA1 P38398 1/20 0.45
CTSC P53634 11/20 0.44
GAA P10253 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP2C19 P33261 1/20 0.43
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DPP4 P27487 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
DPP9 Q86TI2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
CTSL P07711 1/20 0.38
CTSS P25774 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27268932 0.80 PKM (0.51) GAASMN1; SMN2DPP4ALDH1A1
SCHEMBL7301262 0.79 DPP4 (0.40) GLABRCA1GAASMN1; SMN2DPP4
SCHEMBL14191010 0.77 NPC1 (0.47) GLABRCA1GAANPSR1CYP2C19
SCHEMBL1631750 0.75 CTSC (0.59) CTSCCYP2C19RAB9ASLC1A3SLC1A2
SCHEMBL2058609 0.75 CTSC (0.59) CTSCCYP2C19RAB9ASLC1A3SLC1A2
SCHEMBL19699149 0.75 CTSC (0.59) CTSCCYP2C19RAB9ASLC1A3SLC1A2
SCHEMBL6897729 0.74 CYP2C19 (0.53) CTSCCYP2C19RAB9ASLC1A3SLC1A2
SCHEMBL20543720 0.74 CTSC (0.55) CTSCCYP2C19RAB9ANPC1SMN1; SMN2
Hydrochloric Acid SCHEMBL28362983 0.74 CTSC (0.58) CTSCCYP2C19RAB9ASLC1A3SLC1A2
Hydrochloric Acid SCHEMBL2524346 0.74 CTSC (0.58) CTSCCYP2C19RAB9ASLC1A3SLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657453-B1 Angiotensin converting enzyme (ace) inhibitors containing a fused multiple ring lactam BRISTOL MYERS SQUIBB CO (US) 1999-01-20 EP disclosed
US-5637698-A ANGIOTENSIN CONVERTING ENZYME AND NEUTRAL ENDOPEPTIDASE INHIBITOR BRISTOL-MYERS SQUIBB CO. (US) 1997-06-10 US disclosed
US-5525723-A INHIBITORS OF ANGIOTENSIN CONVERTING ENZYME, NEUTRAL ENDOPEPTIDASE BRISTOL-MYERS SQUIBB CO. (US) 1996-06-11 US disclosed
EP-0657453-A1 Angiotensin converting enzyme (ace) inhibitors containing a fused multiple ring lactam BRISTOL-MYERS SQUIBB COMPANY (US) 1995-06-14 EP disclosed