SCHEMBL7307316

SCHEMBL7307316

CCCC[C@H](NC(=O)CC[C@H](C)CNC(=O)COc1ccccc1)C(=O)CS(=O)(=O)Cc1ccco1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.41
PKM P14618 1/20 0.41
POLB P06746 4/20 0.41
MAPT P10636 5/20 0.40
HPGD P15428 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
USP2 O75604 1/20 0.40
MAPK1 P28482 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ESR1 P03372 1/20 0.38
APEX1 P27695 1/20 0.38
TSHR P16473 3/20 0.37
GPR88 Q9GZN0 1/20 0.37
RECQL P46063 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302483 0.85 ALDH1A1 (0.51) ALDH1A1PKMPOLBMAPTHPGD
SCHEMBL7307309 0.84 CASP3 (0.45) ALDH1A1PKMPOLBMAPTHPGD
SCHEMBL7307297 0.84 CASP3 (0.45) ALDH1A1PKMPOLBMAPTHPGD
SCHEMBL7313905 0.84 PKM (0.41) ALDH1A1PKMPOLBMAPTHPGD
SCHEMBL7307300 0.83 TSHR (0.45) ALDH1A1PKMPOLBMAPTHPGD
SCHEMBL7311218 0.80 ALDH1A1 (0.52) ALDH1A1PKMPOLBMAPTHPGD
SCHEMBL7301647 0.76 ALDH1A1 (0.51) ALDH1A1POLBMAPTHPGDTDP1
SCHEMBL7307305 0.75 MAPT (0.36) ALDH1A1PKMPOLBMAPTHPGD
SCHEMBL7303805 0.75 ALDH1A1 (0.52) ALDH1A1POLBMAPTHPGDTDP1
SCHEMBL7315659 0.73 ALDH1A1 (0.54) ALDH1A1POLBMAPTHPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed
EP-0525420-A1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors Mitsubishi Chemical Corporation (JP) 1993-02-03 EP disclosed