SCHEMBL7308066

SCHEMBL7308066

CCOC(=O)[C@@H](NCc1ccc(Br)nc1)C(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.42
MMP2 P08253 2/20 0.41
MMP9 P14780 2/20 0.41
MMP8 P22894 2/20 0.41
MMP13 P45452 2/20 0.41
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGB1 P05556 1/20 0.37
ITGAV P06756 1/20 0.37
ITGA5 P08648 1/20 0.37
MEP1B Q16820 2/20 0.36
CD274 Q9NZQ7 3/20 0.36
PDCD1 Q15116 2/20 0.36
ADRB2 P07550 2/20 0.35
ADRB1 P08588 2/20 0.35
ADRB3 P13945 2/20 0.35
CPB2 Q96IY4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308075 1.00 SIRT2 (0.42) SIRT2MMP2MMP9MMP8MMP13
SCHEMBL21125254 0.90 SIRT2 (0.48) SIRT2MMP2MMP9MMP8MMP13
SCHEMBL7302440 0.74 SIRT2 (0.54) SIRT2MMP2MMP9MMP8MMP13
SCHEMBL7302451 0.74 SIRT2 (0.54) SIRT2MMP2MMP9MMP8MMP13
SCHEMBL16838929 0.73 LTA4H (0.46) ALDH1A1MAPTCD274
SCHEMBL1616321 0.72 ALDH1A1 (0.51) MMP13ALDH1A1MEP1B
SCHEMBL1525379 0.72 MAOB (0.45) LMNAMAPT
SCHEMBL22775570 0.72 TACR1 (0.45) SIRT2ITGB3CPB2
SCHEMBL29605170 0.72 TACR1 (0.45) SIRT2ITGB3CPB2
SCHEMBL2443868 0.71 GAA (0.51) ALDH1A1TDP1ITGB3ITGB1ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5594010-A TREATMENT OF HYPERTENSION AND ATHERIOSCLEROSIS BAYER AKTIENGESELLSCHAFT (DE) 1997-01-14 US disclosed
EP-0630896-A1 Substituted mono- and bipyridylmethyl derivatives as angiotensin II antagonist BAYER AG (DE) 1994-12-28 EP disclosed