SCHEMBL7310468

SCHEMBL7310468

CSCC[C@@H](C(N)=O)N(C)Cc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
SLC6A2 P23975 1/20 0.41
HTR2A P28223 1/20 0.41
SLC6A4 P31645 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRK1 P41145 1/20 0.41
SLC6A3 Q01959 1/20 0.41
KCNH2 Q12809 1/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
ANPEP P15144 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ATM Q13315 1/20 0.39
HPGD P15428 1/20 0.39
AOC3 Q16853 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9081277 0.88 NPC1 (0.42) NPC1RAB9AADRA2BADRA2CSLC6A2
SCHEMBL11095434 0.84 SIGMAR1 (0.46) AOC3
SCHEMBL8086805 0.82 HTR2A (0.41) HTR2AAOC3
SCHEMBL25382623 0.81 CNR2 (0.44) NPC1RAB9AADRA2BADRA2CSLC6A2
SCHEMBL7466902 0.80 NPC1 (0.46) NPC1RAB9AADRA2BADRA2CSLC6A2
SCHEMBL17559642 0.80 NPC1 (0.46) NPC1RAB9AADRA2BADRA2CSLC6A2
SCHEMBL900942 0.80 ADRA2B (0.54) NPC1RAB9AADRA2BADRA2CSLC6A2
SCHEMBL17161709 0.80 NPC1 (0.46) NPC1RAB9AADRA2BADRA2CSLC6A2
SCHEMBL6681598 0.78 ANPEP (0.42) NPC1RAB9ACA12CA9ANPEP
SCHEMBL27768608 0.78 ANPEP (0.42) NPC1RAB9ACA12CA9ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed