SCHEMBL7310609

SCHEMBL7310609

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(OCCn2ccnc2)cc1)C(O)CNC[C@@H](O)[C@H](Cc1ccccc1)NC(=O)O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.49
LTA4H P09960 1/20 0.48
KMT2A Q03164 2/20 0.48
TBXAS1 P24557 12/20 0.47
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
LMNA P02545 2/20 0.43
MEN1 O00255 1/20 0.43
KLK5 Q9Y337 1/20 0.43
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302660 0.84 KLK5 (0.51) CTSSCTSKKLK5
SCHEMBL8955018 0.84 KLK5 (0.46) LMNAKLK5
SCHEMBL7307304 0.83 KLK5 (0.52) KLK5
SCHEMBL7314764 0.83 KLK5 (0.52) KLK5
SCHEMBL8955028 0.82 KLK5 (0.52) KMT2ALMNAMEN1KLK5
SCHEMBL7309371 0.82 KLK5 (0.46) KLK5
SCHEMBL7312642 0.82 KLK5 (0.52) LTA4HKLK5
SCHEMBL8955074 0.81 BACE1 (0.44) KLK5
SCHEMBL7311526 0.81 KLK5 (0.55) KLK5
SCHEMBL7303561 0.81 KLK5 (0.61) CTSSCTSKKLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559256-A Aminediol protease inhibitors E. R. SQUIBB & SONS, INC. (US) 1996-09-24 US disclosed
EP-0580402-A2 Aminediol protease inhibitors E.R. SQUIBB & SONS, INC. (US) 1994-01-26 EP disclosed