SCHEMBL8955018

SCHEMBL8955018

CC(C)(C)OC(=O)N[C@@H](Cc1ccc(OCCOc2cccnc2)cc1)C(O)CNC[C@@H](O)[C@H](Cc1ccccc1)NC(=O)O

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.46
ATM Q13315 1/20 0.43
CYP3A4 P08684 5/20 0.42
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
FAAH O00519 1/20 0.42
PSEN1 P49768 4/20 0.41
PSEN2 P49810 4/20 0.41
APH1B Q8WW43 4/20 0.41
NCSTN Q92542 4/20 0.41
APH1A Q96BI3 4/20 0.41
PSENEN Q9NZ42 4/20 0.41
LMNA P02545 1/20 0.41
BCHE P06276 1/20 0.40
REN P00797 1/20 0.40
BACE1 P56817 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8955096 0.88 KLK5 (0.44) KLK5ATMCYP3A4BCHEREN
SCHEMBL7314764 0.88 KLK5 (0.52) KLK5ATMITGB3ITGA2BPSEN1
SCHEMBL7307304 0.88 KLK5 (0.52) KLK5ATMITGB3ITGA2BPSEN1
SCHEMBL7302660 0.87 KLK5 (0.51) KLK5ATMITGB3ITGA2BPSEN1
SCHEMBL8955028 0.85 KLK5 (0.52) KLK5ATMITGB3ITGA2BPSEN1
SCHEMBL7309371 0.85 KLK5 (0.46) KLK5ATMITGB3ITGA2BPSEN1
SCHEMBL7312642 0.85 KLK5 (0.52) KLK5ATMPSEN1PSEN2APH1B
SCHEMBL8955077 0.84 KLK5 (0.49) KLK5ATMITGB3ITGA2BPSEN1
SCHEMBL7310609 0.84 ACACB (0.49) KLK5LMNA
SCHEMBL7311526 0.84 KLK5 (0.55) KLK5ATMPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5559256-A Aminediol protease inhibitors E. R. SQUIBB & SONS, INC. (US) 1996-09-24 US disclosed