SCHEMBL7310668

SCHEMBL7310668

CS(=O)(=O)OCC1CN(CCCCN2CCN(Cc3ccccc3)CC2)C(=O)O1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
CCR3 P51677 1/20 0.43
HTR7 P34969 2/20 0.42
ALDH1A1 P00352 1/20 0.41
ACHE P22303 1/20 0.41
HTR1A P08908 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308886 0.98 MAPK1 (0.49) MAPK1L3MBTL1CCR3HTR7ALDH1A1
SCHEMBL7305380 0.94 MAPK1 (0.46) MAPK1L3MBTL1HTR7ALDH1A1
SCHEMBL7311493 0.89 MAPK1 (0.45) MAPK1L3MBTL1ACHE
SCHEMBL7315459 0.88 MAPK1 (0.46) MAPK1L3MBTL1ACHE
SCHEMBL7313926 0.86 ACHE (0.51) MAPK1L3MBTL1ACHE
SCHEMBL7306386 0.84 MAPK1 (0.47) MAPK1L3MBTL1
SCHEMBL7315671 0.84 F10 (0.42) CCR3
SCHEMBL8858076 0.83 MAPK1 (0.38) MAPK1L3MBTL1ALDH1A1
SCHEMBL8858183 0.82 HTR2B (0.37) MAPK1L3MBTL1ALDH1A1HTR1A
SCHEMBL8858178 0.82 MEN1 (0.41) L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed