SCHEMBL7305380

SCHEMBL7305380

CS(=O)(=O)OCC1CN(CCN2CCN(Cc3ccccc3)CC2)C(=O)O1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MC4R P32245 1/20 0.40
ALDH1A1 P00352 3/20 0.40
MAPT P10636 1/20 0.40
CCR2 P41597 1/20 0.40
TSHR P16473 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SIGMAR1 Q99720 2/20 0.39
ABCB1 P08183 1/20 0.39
HTR7 P34969 1/20 0.38
RECQL P46063 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GRM2 Q14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7308886 0.94 MAPK1 (0.49) MAPK1L3MBTL1ALDH1A1HTR7
SCHEMBL7310668 0.94 MAPK1 (0.49) MAPK1L3MBTL1ALDH1A1HTR7
SCHEMBL7313926 0.88 ACHE (0.51) MAPK1L3MBTL1
SCHEMBL7315459 0.86 MAPK1 (0.46) MAPK1L3MBTL1
SCHEMBL7315671 0.85 F10 (0.42) SIGMAR1RECQLSMN1; SMN2
SCHEMBL7311493 0.85 MAPK1 (0.45) MAPK1L3MBTL1
SCHEMBL7305151 0.84 MAPK1 (0.39) MAPK1L3MBTL1
SCHEMBL8858127 0.82 HTR2B (0.37) MAPK1L3MBTL1ALDH1A1TSHRSIGMAR1
SCHEMBL8858111 0.81 LMNA (0.41) L3MBTL1ALDH1A1MEN1KMT2ASIGMAR1
SCHEMBL7310189 0.81 RECQL (0.48) ALDH1A1RECQLSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed