SCHEMBL7310995

SCHEMBL7310995

CCCc1nc(C(=O)OCc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)c(CO)n1CC

nearest known ligand 0.50

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 11/20 0.50
AGTR2 P50052 11/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669230 0.90 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL5366890 0.88 AGTR1 (0.49) AGTR1AGTR2
SCHEMBL7302940 0.88 AGTR1 (0.48) AGTR1AGTR2
Hydrochloric Acid SCHEMBL7305271 0.88 AGTR1 (0.48) AGTR1AGTR2
SCHEMBL669265 0.86 AGTR2 (0.52) AGTR1AGTR2
SCHEMBL7304493 0.86 AGTR1 (0.47) AGTR1AGTR2
SCHEMBL3841095 0.83 AGTR2 (0.58) AGTR1AGTR2
SCHEMBL3844504 0.83 AGTR1 (0.46) AGTR1AGTR2
SCHEMBL7886348 0.83 AGTR1 (0.41) AGTR1AGTR2
SCHEMBL7307299 0.83 AGTR1 (0.49) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0545912-B1 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2001-04-25 EP disclosed
US-5646171-A HYPOTENSIVE AGENTS SANKYO COMPANY, LIMITED (JP) 1997-07-08 US disclosed
US-5616599-A HYPOTENSIVE AGENTS FOR CARDIOVASCULAR DISORDER SANKYO COMPANY, LIMITED (JP) 1997-04-01 US disclosed
EP-0545912-A2 1-Biphenylmethylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1993-06-09 EP disclosed
EP-0503785-A1 1-Biphenylimidazole derivatives, their preparation and their therapeutic use Sankyo Company Limited (JP) 1992-09-16 EP disclosed