SCHEMBL7311682

SCHEMBL7311682

COc1ccc(S(=O)(=O)c2c(C(=O)O)cc(C)c(NCc3cccnc3)c2-c2ccco2)cc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 3/20 0.49
MMP9 P14780 3/20 0.49
MMP13 P45452 3/20 0.49
ADAM17 P78536 3/20 0.49
NAMPT P43490 12/20 0.47
ALDH1A1 P00352 3/20 0.46
PKM P14618 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323020 0.94 MMP1 (0.49) MMP1MMP9MMP13ADAM17NAMPT
SCHEMBL7323617 0.92 MMP9 (0.57) MMP1MMP9MMP13ADAM17NAMPT
SCHEMBL7325342 0.75 NAMPT (0.56) MMP1MMP9MMP13ADAM17NAMPT
SCHEMBL7352965 0.74 MMP9 (0.44) MMP1MMP9MMP13ADAM17NAMPT
SCHEMBL7322218 0.74 NAMPT (0.55) MMP1MMP9MMP13NAMPTALDH1A1
SCHEMBL7352954 0.72 KAT6A (0.40) MMP1MMP9MMP13ADAM17ALDH1A1
SCHEMBL7324688 0.72 MMP1 (0.46) MMP1MMP9MMP13ADAM17NAMPT
SCHEMBL7352961 0.71 MMP13 (0.68) MMP1MMP9MMP13ADAM17
SCHEMBL7316683 0.71 NAMPT (0.52) MMP1MMP9MMP13ADAM17NAMPT
SCHEMBL7316583 0.71 NAMPT (0.53) MMP1MMP9MMP13ADAM17NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929097-A INHIBIT TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME AMERICAN CYANAMID COMPANY (US) 1999-07-27 US disclosed