SCHEMBL7312137

SCHEMBL7312137

COc1ccc(C#Cc2ccc(C(F)(F)F)cc2)c(CC(C)N(C)CCc2ccc(OC)c(OC)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.40
AOC3 Q16853 2/20 0.39
CYP3A4 P08684 6/20 0.39
ABCB1 P08183 5/20 0.39
ABCC1 P33527 4/20 0.39
CYP2C19 P33261 3/20 0.39
CYP2D6 P10635 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
CACNA1C Q13936 2/20 0.39
CYP1A2 P05177 2/20 0.39
ABCB11 O95342 2/20 0.39
KCNH2 Q12809 2/20 0.39
TSHR P16473 2/20 0.39
LMNA P02545 2/20 0.39
HTR2A P28223 2/20 0.39
HTR2C P28335 2/20 0.39
HTR2B P41595 2/20 0.39
CYP2C9 P11712 2/20 0.39
SLC22A1 O15245 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7318305 0.88 SMPD1 (0.43) ACACBAOC3CYP3A4CYP2D6MEN1
SCHEMBL9218599 0.80 CYP1A2 (0.41) AOC3CYP3A4CYP2D6MEN1KMT2A
SCHEMBL10686888 0.79 CYP3A4 (0.40) AOC3CYP3A4ABCB1ABCC1CYP2C19
Hydrochloric Acid SCHEMBL7311252 0.79 BLM (0.42) AOC3CYP3A4CYP2D6MEN1KMT2A
Hydrochloric Acid SCHEMBL7349845 0.78 MEN1 (0.43) ACACBCYP3A4CYP2D6MEN1KMT2A
SCHEMBL10688197 0.78 KMT2A (0.41) AOC3CYP3A4CYP2D6MEN1KMT2A
SCHEMBL10738517 0.77 SIGMAR1 (0.42) ACACBAOC3KCNH2
SCHEMBL7316655 0.76 SIGMAR1 (0.42) ACACBMEN1KMT2AKCNH2HTR2A
SCHEMBL10687447 0.76 CYP3A4 (0.49) AOC3CYP3A4CYP2C19CYP2D6MEN1
Oxalic Acid SCHEMBL7318269 0.75 PTGES (0.46) ACACBMEN1KMT2ATSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4742084-A Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives MCNEILAB, INC. (US) 1988-05-03 US disclosed
US-4661635-A ANTIARRHYTHMIA AGENTS MCNEILAB, INC. (US) 1987-04-28 US disclosed
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed