SCHEMBL7316655

SCHEMBL7316655

COc1ccc(C#Cc2ccccc2)c(CC(C)N(C)CCc2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.42
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
GRIN2C Q14957 1/20 0.42
GRIN3A Q8TCU5 1/20 0.42
ACACB O00763 4/20 0.42
MAOB P27338 5/20 0.41
MAOA P21397 1/20 0.41
KCNH2 Q12809 2/20 0.38
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR2A P28223 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7318305 0.88 SMPD1 (0.43) SIGMAR1ACACBMEN1KMT2AHTR2A
SCHEMBL10738517 0.87 SIGMAR1 (0.42) SIGMAR1ACACBMAOBMAOAKCNH2
Hydrochloric Acid SCHEMBL7312601 0.82 SIGMAR1 (0.51) SIGMAR1MAOB
SCHEMBL10411872 0.79 MTNR1A (0.40) SIGMAR1ACACBMAOBMAOA
SCHEMBL9218599 0.79 CYP1A2 (0.41) SIGMAR1MEN1KMT2AHTR2A
Hydrochloric Acid SCHEMBL7311252 0.79 BLM (0.42) SIGMAR1MEN1KMT2AHTR2A
Hydrochloric Acid SCHEMBL7349845 0.77 MEN1 (0.43) ACACBMAOBKCNH2MEN1KMT2A
SCHEMBL7312137 0.76 ACACB (0.40) ACACBKCNH2MEN1KMT2AHTR2A
Oxalic Acid SCHEMBL7318269 0.74 PTGES (0.46) ACACBMAOBMEN1KMT2A
SCHEMBL10411855 0.73 MTNR1A (0.44) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4742084-A Aralykyl (arylethynyl)aralkyl amines and their use as vasodilators and antihypertensives MCNEILAB, INC. (US) 1988-05-03 US disclosed
US-4661635-A ANTIARRHYTHMIA AGENTS MCNEILAB, INC. (US) 1987-04-28 US disclosed
EP-0146271-A2 Aralykyl (arylethynyl) aralkyl amines for use as vasodilators and antihypertensives McNeilab, Inc. (US) 1985-06-26 EP disclosed