SCHEMBL7313642

SCHEMBL7313642

CCOc1[c]c(CBr)ccc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.33
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
ELANE P08246 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LTA4H P09960 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7314203 0.85 KMT2A (0.33) LTA4H
SCHEMBL7772526 0.84 NQO1 (0.36) NQO1TP53CYP3A4ALDH1A1LTA4H
SCHEMBL128399 0.81 NQO1 (0.43) NQO1TP53CYP3A4ALDH1A1LTA4H
SCHEMBL7312733 0.80 SMN1; SMN2 (0.32) ALDH1A1
SCHEMBL11503774 0.78 KCNH2 (0.32) NQO1TP53CYP3A4LTA4H
SCHEMBL3362979 0.77 GABRA1 (0.33) NQO1TP53CYP3A4ALDH1A1
SCHEMBL7768476 0.76 NQO1 (0.36) NQO1TP53CYP3A4ALDH1A1LTA4H
SCHEMBL743598 0.74 SMN1; SMN2 (0.38) NQO1TP53CYP3A4ALDH1A1LTA4H
SCHEMBL2962480 0.74 NQO1 (0.37) NQO1TP53CYP3A4ALDH1A1LTA4H
SCHEMBL11612858 0.73 TRPA1 (0.36) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0634396-B1 Amino acid derivatives and their use as inhibitors of encephalinase BIOPROJET SOC CIV (FR) 1998-10-28 EP disclosed
EP-0634396-A1 Amino acid derivatives and their use as inhibitors of encephalinase SOCIETE CIVILE BIOPROJET (FR) 1995-01-18 EP disclosed