SCHEMBL7315480

SCHEMBL7315480

CC(=O)NC1CCc2nc(NC(=O)c3ccccc3)sc2C1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.58
CSNK2A1 P68400 2/20 0.58
GAA P10253 1/20 0.53
TP53 P04637 4/20 0.53
LMNA P02545 3/20 0.51
MAPT P10636 2/20 0.51
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 1/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7312903 0.84 NPC1 (0.54) GSK3BCSNK2A1TP53MAPTRAB9A
SCHEMBL7321908 0.84 MAPT (0.70) GSK3BCSNK2A1TP53LMNAMAPT
SCHEMBL7322371 0.81 MAPT (0.53) GSK3BCSNK2A1TP53LMNAMAPT
Hydrochloric Acid SCHEMBL7323627 0.80 ROCK2 (0.63) GAATP53
SCHEMBL12804931 0.80 NPC1 (0.52) GSK3BCSNK2A1RAB9ANPC1
SCHEMBL3562146 0.80 NPC1 (0.52) GSK3BCSNK2A1RAB9ANPC1
SCHEMBL3562143 0.80 NPC1 (0.52) GSK3BCSNK2A1RAB9ANPC1
SCHEMBL7318633 0.80 SCN3A (0.48) GSK3BCSNK2A1TP53MAPTRAB9A
SCHEMBL7319478 0.80 NPC1 (0.48) GSK3BCSNK2A1RAB9ANPC1
SCHEMBL7324759 0.79 NPC1 (0.52) GSK3BCSNK2A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4886812-A REGULATING DOPAMINE CONCENTRATION; PARKINSON DISEASE, HYPOTENSIVE AGENT, SCHIZOPHRENIA DR. KARL THOMAE GMBH (DE) 1989-12-12 US disclosed
US-4843086-A HYPOTENSIVE AGENTS, SCHIZOPHRENIA, PARKINSON'S DISEASE BOEHRINGER INGELHEIM KG (DE) 1989-06-27 US disclosed
US-4731374-A PARKINSON*S DISEASE DR. KARL THOMAE GMBH (DE) 1988-03-15 US disclosed
EP-0186087-A1 Tetrahydro-benzothiazoles, their production and their use as intermediates or drugs Dr. Karl Thomae GmbH (DE) 1986-07-02 EP disclosed