SCHEMBL7315657

SCHEMBL7315657

COc1cccc(C2(O)c3ccccc3-c3ccccc32)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 4/20 0.51
SCN9A Q15858 1/20 0.48
MEN1 O00255 1/20 0.47
GAA P10253 1/20 0.47
KMT2A Q03164 1/20 0.47
OPRM1 P35372 2/20 0.45
OPRD1 P41143 1/20 0.45
OPRK1 P41145 1/20 0.45
OPRL1 P41146 1/20 0.45
KDM1A O60341 1/20 0.44
SLC6A2 P23975 2/20 0.42
CHRNA1 P02708 1/20 0.42
CHRNG P07510 1/20 0.42
CHRNB1 P11230 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CHRND Q07001 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17439398 0.84 PDK2 (0.64) PDK2MEN1GAAKMT2ASLC6A3
SCHEMBL7324013 0.84 PDK2 (0.60) PDK2MEN1GAAKMT2A
SCHEMBL17456241 0.84 PDK2 (0.52) PDK2MEN1GAAKMT2ASLC6A2
SCHEMBL14191205 0.83 ESR1 (0.47) PDK2SCN9AMEN1GAAKMT2A
SCHEMBL23996970 0.82 PDK2 (0.45) PDK2MEN1KMT2AOPRK1
SCHEMBL15836744 0.81 PDK2 (0.40) PDK2SCN9AMEN1GAAKMT2A
SCHEMBL7315127 0.81 PDK2 (0.51) PDK2SCN9AMEN1GAAKMT2A
SCHEMBL14584274 0.80 ESR1 (0.45) PDK2MEN1KMT2AOPRM1OPRD1
SCHEMBL30829201 0.78 PDK2 (0.57) PDK2MEN1GAAKMT2AALDH1A1
SCHEMBL27392537 0.78 PDK2 (0.57) PDK2MEN1GAAKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6162824-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ALLELIX NEUROSCIENCE INC. 2000-12-19 US disclosed
EP-0975600-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTITHROMBOTIC AGENTS Akzo Nobel N.V. (NL) 2000-02-02 EP disclosed
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO disclosed
WO-1998047876-A1 HETEROCYCLIC DERIVATIVES AND THEIR USE AS ANTITHROMBOTIC AGENTS AKZO NOBEL N.V. (NL) 1998-10-29 WO disclosed
US-5447960-A Fungicidal use of phenolic aromatic compounds DOWELANCO (US) 1995-09-05 US disclosed