SCHEMBL7315909

SCHEMBL7315909

COC(=O)C1=C(C)NC(C)=C(c2nc(CN3CCCCC3)no2)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 4/20 0.57
MAPT P10636 4/20 0.54
ADRA1A P35348 4/20 0.54
HIF1A Q16665 3/20 0.54
MEN1 O00255 3/20 0.54
CYP1A2 P05177 3/20 0.54
CYP3A4 P08684 3/20 0.54
CYP2C9 P11712 3/20 0.54
CYP2C19 P33261 3/20 0.54
KMT2A Q03164 3/20 0.54
ADRA2A P08913 3/20 0.54
ADORA3 P0DMS8 3/20 0.54
CHRM2 P08172 2/20 0.54
HTR1A P08908 2/20 0.54
DRD1 P21728 2/20 0.54
SLC6A2 P23975 2/20 0.54
SLC6A4 P31645 2/20 0.54
OPRM1 P35372 2/20 0.54
DRD3 P35462 2/20 0.54
SLC6A3 Q01959 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10368230 0.92 ABCB1 (0.48) ABCB1MAPTADRA1AHIF1AMEN1
SCHEMBL10368228 0.92 ABCB1 (0.48) ABCB1MAPTADRA1AHIF1AMEN1
SCHEMBL10368511 0.89 ABCB1 (0.46) ABCB1MAPTADRA1AHIF1AMEN1
SCHEMBL7317593 0.89 ABCB1 (0.51) ABCB1MAPTADRA1AHIF1AMEN1
SCHEMBL7319281 0.87 ADORA3 (0.47) ABCB1ADRA1AADRA2AADORA3CHRM2
SCHEMBL7311935 0.87 KCNH2 (0.48) ABCB1MAPTADRA1AHIF1AMEN1
SCHEMBL7316659 0.86 MAPT (0.60) ABCB1MAPTADRA1AHIF1AMEN1
SCHEMBL10998252 0.84 MAPT (0.57) ABCB1MAPTADRA1AHIF1AMEN1
SCHEMBL10998756 0.84 MAPT (0.62) ABCB1MAPTHIF1AMEN1CYP1A2
SCHEMBL7313818 0.83 ADRA2A (0.45) ABCB1ADRA1AKMT2AADRA2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0177965-B1 NOVEL OXA- AND THIADIAZOLYL DERIVATIVES AND THEIR USE SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1990-03-21 EP claimed
US-4705786-A Novel oxadiazolyl-1,4-dihydropyridines useful as antihypertensive agents SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1987-11-10 US claimed
EP-0177965-A2 Novel oxa- and thiadiazolyl derivatives and their use SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1986-04-16 EP claimed