SCHEMBL7316593

SCHEMBL7316593

CCn1nnnc1CCCOc1ccc2c(ccc(=O)n2C(C)=O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 7/20 0.38
HDAC1 Q13547 1/20 0.35
PDE3B Q13370 5/20 0.34
PDE3A Q14432 5/20 0.34
POLB P06746 1/20 0.33
P2RY12 Q9H244 1/20 0.33
MEN1 O00255 1/20 0.33
ABCC4 O15439 1/20 0.33
CACNA1F O60840 1/20 0.33
ABCB11 O95342 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
THPO P40225 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7306581 0.89 KCNA5 (0.40) KCNA5HDAC1ALDH1A1CYP1A2CYP3A4
SCHEMBL7311363 0.88 KCNA5 (0.41) KCNA5HDAC1PDE3BPDE3AMEN1
SCHEMBL7313662 0.86 KCNA5 (0.46) KCNA5PDE3BPDE3AP2RY12MEN1
SCHEMBL7312280 0.86 PDE3B (0.46) PDE3BPDE3AP2RY12MEN1ABCC4
SCHEMBL7311398 0.84 HSD11B1 (0.41) KCNA5ALDH1A1LMNAKMT2ASMN1; SMN2
SCHEMBL7315797 0.82 PDE3B (0.54) HDAC1PDE3BPDE3APOLBP2RY12
SCHEMBL7306355 0.81 KCNA5 (0.40) KCNA5HDAC1PDE3BPDE3APOLB
SCHEMBL7317323 0.80 KCNA5 (0.45) KCNA5HDAC1PDE3BPDE3AALDH1A1
SCHEMBL7312406 0.76 PDE3B (0.43) PDE3BPDE3AP2RY12MEN1ABCC4
SCHEMBL7308692 0.74 KCNA5 (0.51) KCNA5PDE3BPDE3AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4277479-A ANTI-ASTHMATIC, HYPOTENSIVE, ANTI-ULCER, ANTIINFLAMMATORY, VASODILATION, ENZYME INHIBITORS, ANTICOAGULANTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1981-07-07 US disclosed