SCHEMBL7317636

SCHEMBL7317636

Cc1nc2ccccn2c(=O)c1CCN1CCC(c2onc3cc(F)ccc23)CC1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.61
HTR1A P08908 3/20 0.61
CYP2D6 P10635 2/20 0.61
TSHR P16473 2/20 0.61
PMP22 Q01453 2/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
KDM4E B2RXH2 1/20 0.61
MEN1 O00255 1/20 0.61
CYP3A4 P08684 1/20 0.61
MAPT P10636 1/20 0.61
PKM P14618 1/20 0.61
HPGD P15428 1/20 0.61
THPO P40225 1/20 0.61
KMT2A Q03164 1/20 0.61
ACHE P22303 2/20 0.56
HTR2A P28223 12/20 0.51
DRD2 P14416 10/20 0.51
ADRA1A P35348 7/20 0.51
ADRA2A P08913 7/20 0.51
ADRA2B P18089 7/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1443153 0.87 DRD2 (0.68) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL1427955 0.86 DRD2 (0.50) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL9050419 0.85 ADRA2A (0.52) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL7701569 0.84 HTR2C (0.61) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL9050924 0.82 DRD2 (0.44) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL9050755 0.82 DRD2 (0.45) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL9491933 0.82 HTR2C (0.61) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL1119172 0.80 DRD2 (0.75) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL5328181 0.80 DRD2 (0.75) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL4616132 0.79 DRD2 (0.53) HTR2CHTR1ACYP2D6TSHRPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0196132-A2 1,2-Benzisoxazol-3-yl and 1,2-benzisothiazol-3-yl derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1986-10-01 EP disclosed