SCHEMBL7318102

SCHEMBL7318102

Nc1nc(Br)cn2c(Br)cnc12

nearest known ligand 0.39

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.39
ADORA2A P29274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19747465 0.81 ADORA1 (0.37) ADORA1ADORA2A
SCHEMBL14431623 0.81 ADORA1 (0.37) ADORA1ADORA2A
SCHEMBL2179685 0.80 AURKA (0.30)
SCHEMBL14536745 0.78 AURKA (0.30)
SCHEMBL19747597 0.78 GABRA1 (0.30)
SCHEMBL25397536 0.76 ADORA1 (0.37) ADORA1ADORA2A
SCHEMBL8240075 0.75 ADORA2A (0.55) ADORA1ADORA2A
SCHEMBL7319030 0.73 IKBKB (0.43)
SCHEMBL8240149 0.72 AURKA (0.41) ADORA2A
SCHEMBL5401158 0.71 TLR7 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5028605-A Antispasmodic, bronchodilators, uterine relaxants, cardiac analeptics, neurosedatives L'UNIVERSITE DE MONTPELLIER I (FR) 1991-07-02 US disclosed
EP-0348392-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY Université Montpellier I (FR) 1990-01-03 EP disclosed
WO-1988004298-A1 8-ALKYLAMINOIMIDAZO[1,2-A]PYRAZINES AND DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1988-06-16 WO disclosed