SCHEMBL7318237

SCHEMBL7318237

C=C(C)OCCOCc1ccccc1OCC(O)CNC(C)(C)Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASR P41180 15/20 0.56
ADRB2 P07550 7/20 0.47
CYP2D6 P10635 4/20 0.47
ADRB3 P13945 3/20 0.47
SLC6A2 P23975 3/20 0.47
SLC6A4 P31645 3/20 0.47
SLC6A3 Q01959 3/20 0.47
KCNH2 Q12809 3/20 0.47
HTR1A P08908 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7319524 0.88 CASR (0.60) CASRADRB2CYP2D6ADRB3SLC6A2
SCHEMBL7318229 0.86 CASR (0.56) CASRADRB2CYP2D6ADRB3SLC6A2
SCHEMBL7319712 0.86 CASR (0.58) CASRADRB2CYP2D6ADRB3SLC6A2
SCHEMBL7319039 0.85 ADRB2 (0.54) ADRB2CYP2D6ADRB3SLC6A2SLC6A4
SCHEMBL7317233 0.83 CASR (0.59) CASRADRB2CYP2D6ADRB3SLC6A2
SCHEMBL7312078 0.83 ADRB2 (0.62) ADRB2CYP2D6ADRB3SLC6A2SLC6A4
SCHEMBL11511416 0.81 CASR (0.59) CASRADRB2CYP2D6ADRB3SLC6A2
SCHEMBL7318971 0.78 ADRB2 (0.50) ADRB2CYP2D6ADRB3SLC6A2SLC6A4
SCHEMBL7307486 0.77 CASR (0.60) CASRADRB2CYP2D6ADRB3SLC6A2
SCHEMBL7307118 0.77 CASR (0.59) CASRADRB2CYP2D6ADRB3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4258062-A ISOPRENALINE ANTAGONISTS EFFECTING HEART RATE AND BLOOD PRESSURE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-03-24 US disclosed
US-4171370-A Phenoxy-amino-propanols MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-10-16 US disclosed