SCHEMBL7318902

SCHEMBL7318902

N#CCCOC1N=C(c2ccccc2)c2cc(Cl)ccc2N(CCC#N)C1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 3/20 0.48
HTR2B P41595 1/20 0.48
OPRK1 P41145 5/20 0.48
LMNA P02545 3/20 0.48
PDE3A Q14432 1/20 0.48
NR1I2 O75469 2/20 0.41
ADORA3 P0DMS8 2/20 0.41
OPRM1 P35372 1/20 0.41
KCNH2 Q12809 2/20 0.41
ALB P02768 2/20 0.41
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
CACNA1F O60840 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
AKR1C3 P42330 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7331934 0.90 OPRK1 (0.49) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL7332842 0.88 CCKBR (0.47) PDE4DHTR2BOPRK1LMNAKCNH2
SCHEMBL7320833 0.84 OPRK1 (0.66) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL25409864 0.82 OPRK1 (0.52) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL31366637 0.82 OPRK1 (0.52) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL25409870 0.82 OPRK1 (0.52) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL25408967 0.79 HDAC3 (0.52) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL31366547 0.79 HDAC3 (0.52) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL25408970 0.79 HDAC3 (0.52) PDE4DHTR2BOPRK1LMNAPDE3A
SCHEMBL25408963 0.79 HDAC3 (0.52) PDE4DHTR2BOPRK1LMNAPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4388313-A Novel 3-hydroxy-1,4-benzodiazepine-2-ones and process for the preparation thereof GEROT-PHARMAZEUTIKA GESELLSCHAFT M.B.H. (AT) 1983-06-14 US disclosed