SCHEMBL7319378

SCHEMBL7319378

O=C(O)CCCCCNC(=NC(=O)OCc1ccccc1)NC(=O)OCc1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.62
TGM2 P21980 1/20 0.50
FOLH1 Q04609 5/20 0.48
KEAP1 Q14145 2/20 0.48
NFE2L2 Q16236 2/20 0.48
PTGER4 P35408 3/20 0.45
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KMT2A Q03164 1/20 0.45
SIRT5 Q9NXA8 1/20 0.45
SIRT2 Q8IXJ6 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
TSHR P16473 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029846 1.00 HTT (0.62) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL14628582 0.99 HTT (0.64) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL7318682 0.99 HTT (0.64) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL14598314 0.99 HTT (0.64) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL7359305 0.95 HTT (0.69) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL989685 0.94 TGM2 (0.55) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL8039590 0.93 HTT (0.52) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL7355388 0.90 HTT (0.57) HTTTGM2FOLH1KEAP1NFE2L2
SCHEMBL7314617 0.90 HTT (0.49) HTTTGM2KEAP1NFE2L2LMNA
SCHEMBL7381045 0.88 HTT (0.50) HTTTGM2FOLH1KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999048911-A1 MONOBACTAM ENZYME INHIBITORS NAEJA PHARMACEUTICAL INC. (GB) 1999-09-30 WO disclosed
EP-0646573-A1 Preparation of protected and unprotected guanidino-substituted carboxylic acids HOECHST AKTIENGESELLSCHAFT (DE) 1995-04-05 EP disclosed
US-5326863-A Antithrombin and antitrypsin activity BRISTOL-MYERS SQUIBB COMPANY (US) 1994-07-05 US disclosed
US-5175283-A Enzyme inhibitors for antitrypsin or antithrombin as anticoagulants BRISTOL-MYERS SQUIBB COMPANY (US) 1992-12-29 US disclosed
US-5110812-A Treatment of pancreatitis; anticoagulants BRISTOL-MYERS SQUIBB CO. (US) 1992-05-05 US disclosed
US-5037819-A Anticoagulant; treating pancreatitis BRISTOL-MYERS SQUIBB COMPANY (US) 1991-08-06 US disclosed