SCHEMBL7319557

SCHEMBL7319557

COC(=O)c1c(Cc2cccnc2)c(-c2ccc(C(C)=O)s2)c(N)c(C)c1S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.42
MMP9 P14780 7/20 0.40
MMP13 P45452 7/20 0.40
MMP1 P03956 6/20 0.40
ADAM17 P78536 5/20 0.39
CISD2 Q8N5K1 1/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7321470 0.93 NAMPT (0.41) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7322011 0.93 MMP9 (0.43) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7322608 0.90 NAMPT (0.42) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7321883 0.87 NAMPT (0.43) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7320893 0.86 NAMPT (0.46) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7324058 0.85 NAMPT (0.49) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7317439 0.83 MMP13 (0.49) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7319145 0.83 NAMPT (0.47) NAMPTMMP9MMP13MMP1ADAM17
SCHEMBL7312212 0.83 NAMPT (0.41) NAMPTMMP9MMP13MMP1KEAP1
SCHEMBL7324688 0.83 MMP1 (0.46) NAMPTMMP9MMP13MMP1ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929097-A INHIBIT TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME AMERICAN CYANAMID COMPANY (US) 1999-07-27 US disclosed