SCHEMBL7320022

SCHEMBL7320022

COc1ccc(CCNCC(O)COc2ccc(COCCOC(C)C)cc2)cc1OC

nearest known ligand 0.78

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.78
KMT2A Q03164 1/20 0.68
ADRB1 P08588 2/20 0.62
ADRB3 P13945 1/20 0.62
HTR1A P08908 1/20 0.62
ADRA2C P18825 1/20 0.62
SLC6A4 P31645 1/20 0.62
ADRA1A P35348 1/20 0.62
HTR2B P41595 1/20 0.62
SLC6A3 Q01959 1/20 0.62
KCNH2 Q12809 1/20 0.62
KDM4E B2RXH2 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317527 0.89 KMT2A (0.67) ADRB2KMT2AADRB1HTR1AADRA2C
SCHEMBL7317203 0.88 KMT2A (0.65) ADRB2KMT2AADRB1HTR1AADRA2C
SCHEMBL7314970 0.87 KMT2A (0.64) ADRB2KMT2AADRB1HTR1AADRA2C
SCHEMBL7311212 0.86 ADRB2 (0.60) ADRB2KMT2AADRB1ADRB3HTR1A
SCHEMBL5963374 0.85 KMT2A (0.72) ADRB2KMT2AADRB1HTR1AADRA2C
SCHEMBL4531206 0.85 KMT2A (0.72) ADRB2KMT2AADRB1HTR1AADRA2C
SCHEMBL7312146 0.85 ADRB3 (0.69) ADRB2KMT2AADRB1ADRB3
SCHEMBL7313756 0.84 KMT2A (0.68) ADRB2KMT2AADRB1HTR1AADRA2C
Hydrochloric Acid SCHEMBL7305120 0.83 KMT2A (0.70) ADRB2KMT2AADRB1HTR1AADRA2C
SCHEMBL8835982 0.82 KMT2A (0.78) ADRB2KMT2AADRB1ADRB3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4258062-A ISOPRENALINE ANTAGONISTS EFFECTING HEART RATE AND BLOOD PRESSURE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1981-03-24 US disclosed
US-4171370-A Phenoxy-amino-propanols MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-10-16 US disclosed