SCHEMBL7320059

SCHEMBL7320059

CC(C)NC(=O)CC(C=O)Cc1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.45
MMP9 P14780 3/20 0.45
MMP8 P22894 2/20 0.45
MMP2 P08253 1/20 0.45
MME P08473 2/20 0.45
ACE P12821 2/20 0.45
CPA1 P15085 1/20 0.45
ACE2 Q9BYF1 1/20 0.45
CTNNB1 P35222 1/20 0.44
MMP14 P50281 1/20 0.43
KMT2A Q03164 1/20 0.43
ATM Q13315 1/20 0.41
LMNA P02545 2/20 0.41
HRH4 Q9H3N8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446875 0.82 CTNNB1 (0.49) MMP9MMEACECPA1ACE2
SCHEMBL6448370 0.81 TDP1 (0.54) CASP1MMEACECPA1ACE2
SCHEMBL7276360 0.80 MMP9 (0.45) MMP9MMP8MMP2MMEACE
SCHEMBL7303541 0.79 CTNNB1 (0.46) CASP1MMP9MMEACECPA1
SCHEMBL8484930 0.79 CTNNB1 (0.51) CTNNB1KMT2A
SCHEMBL10589995 0.78 KMT2A (0.54) CASP1CTNNB1KMT2ALMNA
SCHEMBL7319434 0.78 NPC1 (0.49) MMEACEKMT2ALMNA
SCHEMBL7299907 0.78 ALOX15 (0.46) CASP1MMP9
SCHEMBL2752797 0.78 ATM (0.60) KMT2AATMLMNA
SCHEMBL7294849 0.77 CTNNB1 (0.44) MMP9MMEACECPA1ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0327877-A2 Peptide-renininhibitors MERCK PATENT GmbH (DE) 1989-08-16 EP disclosed
EP-0292800-A2 Amino acid derivatives MERCK PATENT GmbH (DE) 1988-11-30 EP disclosed
EP-0249096-A2 Renin-inhibiting amino acid derivatives MERCK PATENT GmbH (DE) 1987-12-16 EP disclosed