SCHEMBL7299907

SCHEMBL7299907

CN(C)CCCNC(=O)CC(C=O)Cc1cccc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.46
CASP1 P29466 1/20 0.45
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA3 P07451 1/20 0.44
CA4 P22748 1/20 0.44
CA6 P23280 1/20 0.44
CA5A P35218 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
CA5B Q9Y2D0 1/20 0.44
CCR4 P51679 1/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
OPRM1 P35372 2/20 0.41
MMP9 P14780 1/20 0.41
KDM4E B2RXH2 1/20 0.41
HTT P42858 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294460 0.82 ALOX15 (0.54) ALOX15CASP1KDM4EHTT
SCHEMBL10589995 0.81 KMT2A (0.54) CASP1OPRM1MTNR1A
SCHEMBL7302653 0.80 HTR1B (0.43) CYP2C19MMP9
SCHEMBL7294849 0.78 CTNNB1 (0.44) CYP2C19OPRM1MMP9
SCHEMBL7320059 0.78 CASP1 (0.45) CASP1MMP9
SCHEMBL7299772 0.77 ALOX15 (0.49) ALOX15CASP1HTT
SCHEMBL6442868 0.76 MMP9 (0.45) CASP1OPRM1MMP9MTNR1A
SCHEMBL6446875 0.76 CTNNB1 (0.49) MMP9MTNR1A
SCHEMBL6448370 0.74 TDP1 (0.54) CASP1CYP2C9CYP2C19HTT
SCHEMBL9666926 0.74 CYP1A2 (0.47) CYP2C9CYP2C19OPRM1MMP9HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5401722-A Peptide analogues MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-03-28 US disclosed
EP-0501280-A2 Renin-inhibiting peptide analogues MERCK PATENT GmbH (DE) 1992-09-02 EP disclosed
EP-0446485-A2 Peptide analogues with renininhibiting activity MERCK PATENT GmbH (DE) 1991-09-18 EP disclosed
EP-0342325-A2 Renin-inhibiting amino acid derivatives MERCK PATENT GmbH (DE) 1989-11-23 EP disclosed
EP-0339483-A2 Renin inhbiting amino-acid derivatives MERCK PATENT GmbH (DE) 1989-11-02 EP disclosed