SCHEMBL7320568

SCHEMBL7320568

CC(OC1(c2ccccc2F)c2ccccc2-c2ccccc21)[C@H](N)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.38
PDK2 Q15119 4/20 0.38
HCAR2 Q8TDS4 1/20 0.36
CYP1A2 P05177 3/20 0.35
CYP2C19 P33261 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
SLC1A3 P43003 2/20 0.35
SLC1A2 P43004 2/20 0.35
SLC1A1 P43005 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2D6 P10635 1/20 0.35
THRB P10828 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HIF1A Q16665 2/20 0.33
PTGS1 P23219 3/20 0.33
PTGS2 P35354 2/20 0.33
LMNA P02545 2/20 0.33
FABP2 P12104 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7320576 1.00 KIF11 (0.38) KIF11PDK2HCAR2CYP1A2CYP2C19
SCHEMBL7325812 0.85 KIF11 (0.38) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7325808 0.85 KIF11 (0.38) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7317362 0.85 KIF11 (0.44) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7323867 0.85 KIF11 (0.44) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7317367 0.85 KIF11 (0.44) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7323278 0.85 KIF11 (0.49) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7323274 0.85 KIF11 (0.49) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7323246 0.83 KIF11 (0.38) KIF11PDK2CYP1A2CYP2C19MEN1
SCHEMBL7325936 0.83 KMT2A (0.41) KIF11PDK2CYP1A2CYP2C19MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO claimed
US-6162824-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ALLELIX NEUROSCIENCE INC. 2000-12-19 US disclosed
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO disclosed