SCHEMBL7323274

SCHEMBL7323274

CC(OC1(c2ccc(F)cc2)c2ccccc2-c2ccccc21)[C@H](N)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.49
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
PDK2 Q15119 2/20 0.36
HIF1A Q16665 1/20 0.36
SLC1A3 P43003 3/20 0.33
SLC1A2 P43004 3/20 0.33
SLC1A1 P43005 3/20 0.33
MEN1 O00255 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
THRB P10828 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
NPC1 O15118 1/20 0.32
CHRM5 P08912 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7323278 1.00 KIF11 (0.49) KIF11CYP1A2CYP2C19PDK2HIF1A
SCHEMBL7317367 0.91 KIF11 (0.44) KIF11CYP1A2CYP2C19PDK2HIF1A
SCHEMBL7317362 0.91 KIF11 (0.44) KIF11CYP1A2CYP2C19PDK2HIF1A
SCHEMBL7323867 0.91 KIF11 (0.44) KIF11CYP1A2CYP2C19PDK2HIF1A
SCHEMBL7318074 0.88 CYP2C19 (0.49) KIF11CYP1A2CYP2C19PDK2HIF1A
SCHEMBL7318078 0.88 CYP2C19 (0.49) KIF11CYP1A2CYP2C19PDK2HIF1A
SCHEMBL7326219 0.87 KIF11 (0.39) KIF11CYP1A2CYP2C19SLC1A3SLC1A2
SCHEMBL7326222 0.87 KIF11 (0.39) KIF11CYP1A2CYP2C19SLC1A3SLC1A2
SCHEMBL7316115 0.86 KIF11 (0.45) KIF11PDK2SLC1A3SLC1A2SLC1A1
SCHEMBL7316108 0.86 KIF11 (0.45) KIF11PDK2SLC1A3SLC1A2SLC1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO claimed
US-6162824-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ALLELIX NEUROSCIENCE INC. 2000-12-19 US disclosed
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO disclosed