SCHEMBL7322735

SCHEMBL7322735

Cc1cccc(C2(OC(C)[C@H](N)C(=O)O)c3ccccc3Oc3ccccc32)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.36
LMNA P02545 2/20 0.36
HCAR2 Q8TDS4 1/20 0.33
KIF11 P52732 5/20 0.33
HDAC4 P56524 1/20 0.33
SLC6A1 P30531 1/20 0.32
CASR P41180 1/20 0.32
CCR2 P41597 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
EDNRB P24530 1/20 0.32
EDNRA P25101 1/20 0.32
SLC1A3 P43003 1/20 0.31
SLC1A2 P43004 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7322744 1.00 NPSR1 (0.36) NPSR1LMNAHCAR2KIF11HDAC4
SCHEMBL7322674 0.90 SLC6A1 (0.38) KIF11SLC6A1CASRMEN1CYP1A2
SCHEMBL7322679 0.90 SLC6A1 (0.38) KIF11SLC6A1CASRMEN1CYP1A2
SCHEMBL7319255 0.90 SLC6A1 (0.38) KIF11SLC6A1CASRMEN1CYP1A2
SCHEMBL7319245 0.90 SLC6A1 (0.38) KIF11SLC6A1CASRMEN1CYP1A2
SCHEMBL7326219 0.82 KIF11 (0.39) KIF11SLC6A1MEN1CYP1A2CYP2D6
SCHEMBL7326222 0.82 KIF11 (0.39) KIF11SLC6A1MEN1CYP1A2CYP2D6
SCHEMBL7320451 0.80 KIF11 (0.40) NPSR1LMNAHCAR2KIF11SLC6A1
SCHEMBL7322275 0.80 KIF11 (0.40) NPSR1LMNAHCAR2KIF11SLC6A1
SCHEMBL7312848 0.77 KIF11 (0.41) NPSR1LMNAKIF11CASRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO claimed
US-6162824-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ALLELIX NEUROSCIENCE INC. 2000-12-19 US disclosed
WO-1999041227-A1 TRICYCLIC COMPOUNDS AS GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-08-19 WO disclosed