SCHEMBL7322931

SCHEMBL7322931

COc1cc(NC(=O)CCCl)ccc1OCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.63
RAB9A P51151 2/20 0.63
HDAC1 Q13547 5/20 0.61
HDAC2 Q92769 5/20 0.61
CTSV O60911 3/20 0.60
CTSL P07711 3/20 0.60
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
KDM4E B2RXH2 1/20 0.57
MAPT P10636 3/20 0.55
LMNA P02545 2/20 0.55
ALDH1A1 P00352 1/20 0.55
ALOX12 P18054 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HPGD P15428 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
C5AR1 P21730 1/20 0.52
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7327512 0.85 NPC1 (0.63) NPC1RAB9AMEN1KMT2AKDM4E
SCHEMBL9653543 0.82 C5AR1 (0.59) NPC1RAB9AHDAC1HDAC2CTSV
SCHEMBL17372654 0.81 NPC1 (0.60) NPC1RAB9AHDAC1HDAC2CTSV
SCHEMBL7356345 0.80 NPC1 (0.65) NPC1RAB9AHDAC1HDAC2CTSV
SCHEMBL7323568 0.80 CYP3A4 (0.64) NPC1RAB9AHDAC1HDAC2CTSV
SCHEMBL22502390 0.80 C5AR1 (0.62) NPC1RAB9AHDAC1CTSVCTSL
SCHEMBL3241459 0.79 MEN1 (0.81) NPC1RAB9AHDAC1HDAC2CTSV
SCHEMBL832694 0.78 LTA4H (0.65) RAB9ACTSVCTSLMEN1KMT2A
SCHEMBL9653129 0.77 C5AR1 (0.59) NPC1RAB9AHDAC1HDAC2CTSV
SCHEMBL17372673 0.77 NPC1 (0.55) NPC1RAB9AHDAC1HDAC2CTSV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0852142-A1 Diamines in the treatment of arrhythmia SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1998-07-08 EP disclosed
EP-0639973-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1995-03-01 EP disclosed
WO-1993023024-A1 DIAMINES IN THE TREATMENT OF ARRHYTHMIA SMITHKLINE BEECHAM LABORATOIRES PHARMACEUTIQUES (FR) 1993-11-25 WO disclosed