SCHEMBL73231

SCHEMBL73231

CC(=O)ON(C(C)=O)c1ccc2c(c1)Cc1ccccc1-2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.49
HTR2C P28335 2/20 0.49
HTR2B P41595 2/20 0.49
ADRA2A P08913 1/20 0.49
MAOA P21397 1/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A4 P31645 1/20 0.49
SRD5A2 P31213 1/20 0.47
CYP3A4 P08684 3/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
HSD17B10 Q99714 2/20 0.46
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.42
DRD2 P14416 1/20 0.41
ADRA1D P25100 1/20 0.41
HTR2A P28223 1/20 0.41
HTR7 P34969 1/20 0.41
ADRA1A P35348 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7092330 0.81 CYP1A2 (0.55) CYP1A2HTR2CHTR2BADRA2AMAOA
SCHEMBL30184649 0.80 CYP1A2 (0.54) CYP1A2HTR2CHTR2BADRA2AMAOA
SCHEMBL637635 0.80 CYP1A2 (0.54) CYP1A2HTR2CHTR2BADRA2AMAOA
SCHEMBL10708948 0.78 CYP1A2 (0.56) CYP1A2HTR2CHTR2BADRA2AMAOA
Sulfuric Acid SCHEMBL2519209 0.75 CYP1A2 (0.49) CYP1A2HTR2CHTR2BADRA2AMAOA
SCHEMBL3503937 0.75 RAB9A (0.49) CYP1A2HTR2CHTR2BADRA2AMAOA
SCHEMBL2532580 0.73 MEN1 (0.47) CYP1A2CYP2C19RAB9ANPC1KDM4E
SCHEMBL1639476 0.72 CYP1A2 (0.58) CYP1A2HTR2CHTR2BADRA2AMAOA
SCHEMBL17264178 0.72 CYP1A2 (0.58) CYP1A2HTR2CHTR2BADRA2AMAOA
SCHEMBL6536307 0.72 MAPT (0.58) CYP1A2HTR2CHTR2BADRA2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8609419-B2 Method for inserting a nucleic acid of interest into a prokaryotic or eukaryotic cell by homologous recombination CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2013-12-17 US claimed
EP-1556496-B1 METHOD FOR INSERTING A NUCLEIC ACID OF INTEREST INTO A PROKARYOTIC OR EUKARYOTIC CELL BY HOMOLOGOUS RECOMBINATION CENTRE NAT RECH SCIENT (FR) 2007-07-25 EP claimed
US-20060270039-A1 Method for inserting a nucleic acid of interest into a prokaryotic or eukaryotic cell by homologous recombination CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2006-11-30 US claimed
EP-1556496-A2 METHOD FOR INSERTING A NUCLEIC ACID OF INTEREST INTO A PROKARYOTIC OR EUKARYOTIC CELL BY HOMOLOGOUS RECOMBINATION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2005-07-27 EP claimed
WO-2004039983-A2 METHOD FOR INSERTING A NUCLEIC ACID OF INTEREST INTO A PROKARYOTIC OR EUKARYOTIC CELL BY HOMOLOGOUS RECOMBINATION CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2004-05-13 WO claimed
CN-105793434-B DNA sequencing and epigenomic analysis STC.UNM 公司 2021-08-10 CN disclosed
CN-105769931-B Oncolytic rhabdovirus 渥太华医院研究机构 2021-04-27 CN disclosed
US-20200056232-A1 DNA SEQUENCING AND EPIGENOME ANALYSIS STC UNM (US) 2020-02-20 US disclosed
EP-3027775-B1 DNA SEQUENCING AND EPIGENOME ANALYSIS STC UNM (US) 2019-10-09 EP disclosed
US-10329614-B2 DNA sequencing and epigenome analysis STC.UNM (US) 2019-06-25 US disclosed
US-20180187190-A1 NEW CRISPR ASSAYS ERASMUS UNIVERSITY MEDICAL CENTER ROTTERDAM (NL) 2018-07-05 US disclosed
US-20160291024-A1 Biomarkers for Ovarian Cancer THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2016-10-06 US disclosed
WO-1990008838-A1 LABELING OF NUCLEIC ACIDS WITH FLUORESCENT MARKERS RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1990-08-09 WO disclosed
EP-0253894-A1 DNA PROBE AND METHOD OF PREPARING THE SAME TORAY INDUSTRIES, INC. (JP) 1988-01-27 EP disclosed
EP-0251527-A2 Haptenylated reagents and immunoassays Panab Laboratories, Inc. (US) 1988-01-07 EP disclosed
WO-1987004165-A1 DNA PROBE AND METHOD OF PREPARING THE SAME TORAY INDUSTRIES, INC. (JP) 1987-07-16 WO disclosed
EP-0097664-B1 PROCESS INVOLVING A PROBE CONTAINING A MODIFIED NUCLEIC ACID RECOGNIZABLE BY SPECIFIC ANTIBODIES AND ALLOWING TO TEST FOR AND CHARACTERIZE AN HOMOLOGOUS DNA SEQUENCE INSTITUT PASTEUR (FR) 1986-03-12 EP disclosed
EP-0128018-A2 Molecular genetic probe, and method of forming same, assay technique and kit using said molecular genetic probe Orgenics Ltd. (IL) 1984-12-12 EP disclosed
US-4469786-A FRAMESHIFT AS WELL AS BASE SUBSTITUTION MUTATIONS THE MOUNT SINAI SCHOOL OF MEDICINE OF THE CITY UNIVERSITY OF NEW YORK (US) 1984-09-04 US disclosed
US-4066510-A ASSAY FOR MUTAGENESIS IN DIPLOID HUMAN LYMPHOBLASTS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1978-01-03 US disclosed